SCHEMBL5147632

SCHEMBL5147632

CCOC(=O)[C@H](Cc1ccc(Oc2nc(C)cc3ccncc23)cc1)NC1=CC(=O)C12CCCCC2

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 13/20 0.46
ITGB1 P05556 12/20 0.46
ELANE P08246 1/20 0.34
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
NLRP3 Q96P20 1/20 0.32
MAPT P10636 1/20 0.30
ITGB7 P26010 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2973969 0.92 ITGA4 (0.54) ITGA4ITGB1CYP3A4CYP2C9ITGB7
SCHEMBL5575858 0.92 ITGA4 (0.54) ITGA4ITGB1CYP3A4CYP2C9ITGB7
SCHEMBL5148508 0.91 ITGB1 (0.47) ITGA4ITGB1ELANECYP3A4CYP2C9
SCHEMBL3830571 0.87 ITGB1 (0.46) ITGA4ITGB1CYP3A4CYP2C9
SCHEMBL3835880 0.86 ITGB1 (0.46) ITGA4ITGB1ELANECYP3A4CYP2C9
SCHEMBL5147636 0.81 ITGB1 (0.38) ITGA4ITGB1
SCHEMBL2974021 0.81 ITGB1 (0.54) ITGA4ITGB1CYP3A4CYP2C9
SCHEMBL7265369 0.81 ITGB1 (0.54) ITGA4ITGB1CYP3A4CYP2C9
SCHEMBL5147640 0.80 ITGB1 (0.35) ITGA4ITGB1MAPT
SCHEMBL3832796 0.80 ITGB1 (0.47) ITGA4ITGB1ELANECYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070167483-A1 2-[(2-Isopropylsulfanyl-3-oxo-spiro[3.5]non-1-en-1-yl)amino]-3-[4-([2,7]naphthyridin-1-ylamino)phenyl]propanoic acid; compounds can inhibit the binding of integrins to their ligands and are of use in the prophylaxis and treatment of immuno or inflammatory disorders UCB PHARMA S.A. (BE) 2007-07-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070167483-A1 2-[(2-Isopropylsulfanyl-3-oxo-spiro[3.5]non-1-en-1-yl)amino]-3-[4-([2,7]naphthyridin-1-ylamino)phenyl]propanoic acid; compounds can inhibit the binding of integrins to their ligands and are of use in the prophylaxis and treatment of immuno or inflammatory disorders ITGB2, VCAM1, ITGB1 ITGA4 40/4885ITGB1 3/4885ELANE 275/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.