SCHEMBL5149159

SCHEMBL5149159

CS(=O)(=O)c1ccc(-c2cc(CO)nn2Cc2ccccc2)cc1

nearest known ligand 0.66

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 9/20 0.66
PTGS1 P23219 4/20 0.53
CA1 P00915 3/20 0.51
CA2 P00918 3/20 0.51
CA9 Q16790 3/20 0.51
SLC16A3 O15427 2/20 0.49
SLC16A1 P53985 1/20 0.48
MCTS1 Q9ULC4 1/20 0.48
ALOX5 P09917 1/20 0.47
HSP90AA1 P07900 1/20 0.47
HSP90B1 P14625 1/20 0.47
TRAP1 Q12931 1/20 0.47
MALT1 Q9UDY8 1/20 0.46
FYN P06241 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2225688 0.85 SLC16A3 (0.59) PTGS2CA1CA2CA9SLC16A3
SCHEMBL4964542 0.82 PTGS2 (0.60) PTGS2PTGS1SLC16A3SLC16A1MCTS1
SCHEMBL3864236 0.82 PTGS2 (0.90) PTGS2PTGS1CA1CA2CA9
SCHEMBL4958833 0.80 MALT1 (0.56) PTGS2PTGS1SLC16A3SLC16A1MCTS1
SCHEMBL9941289 0.80 PTGS2 (1.00) PTGS2PTGS1CA1CA2CA9
SCHEMBL18301051 0.76 SLC16A3 (0.65) PTGS2SLC16A3SLC16A1MCTS1MALT1
SCHEMBL4960172 0.76 PTGS2 (0.52) PTGS2PTGS1CA1CA2CA9
SCHEMBL3867856 0.75 PTGS2 (0.78) PTGS2PTGS1CA1CA2CA9
SCHEMBL3940435 0.74 PTGS2 (0.61) PTGS2PTGS1
SCHEMBL3869730 0.73 CA1 (0.80) PTGS2PTGS1CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7244753-B2 Cyclooxygenase-2 selective inhibitors, compositions and methods of use NITROMED, INC. (US) 2007-07-17 US claimed
US-20040072883-A1 Cyclooxygenase-2 selective inhibitors, compositions and methods of use NITROMED, INC. 2004-04-15 US claimed
US-20070238735-A1 Cyclooxygenase-2 selective inhibitors, compositions and methods of use NITRODMED, INC. (US) 2007-10-11 US disclosed
US-7244753-B2 Cyclooxygenase-2 selective inhibitors, compositions and methods of use NITROMED, INC. (US) 2007-07-17 US disclosed
US-20040072883-A1 Cyclooxygenase-2 selective inhibitors, compositions and methods of use NITROMED, INC. 2004-04-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040072883-A1 Cyclooxygenase-2 selective inhibitors, compositions and methods of use PTGS2, PTGIS, PTGES2 PTGS2 1/4885PTGS1 4/4885CA1 3581/4885
US-20070238735-A1 Cyclooxygenase-2 selective inhibitors, compositions and methods of use PTGS2, PTGIS, PTGS1 PTGS2 1/4885PTGS1 3/4885CA1 3675/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.