SCHEMBL5149869

SCHEMBL5149869

Nc1cccc(Br)c1NC(=O)C[Fe]

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 7/20 0.37
HDAC3 O15379 6/20 0.37
HDAC2 Q92769 5/20 0.37
HDAC10 Q969S8 4/20 0.37
HDAC6 Q9UBN7 4/20 0.37
HDAC4 P56524 4/20 0.37
HDAC7 Q8WUI4 3/20 0.37
HDAC11 Q96DB2 3/20 0.37
HDAC8 Q9BY41 3/20 0.37
HDAC9 Q9UKV0 3/20 0.37
HDAC5 Q9UQL6 3/20 0.37
NCOR2 Q9Y618 2/20 0.37
KMT2A Q03164 3/20 0.36
ALDH1A1 P00352 2/20 0.36
MAPK1 P28482 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4628755 0.79 HDAC1 (0.48) HDAC1HDAC3HDAC2ALDH1A1CA12
SCHEMBL5149864 0.77 HDAC1 (0.47) HDAC1HDAC3HDAC2ALDH1A1CA12
SCHEMBL21684713 0.75 ADORA3 (0.48) HDAC3NCOR2ALDH1A1L3MBTL1
SCHEMBL12948524 0.72 PRKCI (0.34) HDAC1HDAC3MAPK13MAPK12MAPK11
SCHEMBL10750818 0.72 ALDH1A1 (0.42) HDAC1HDAC3HDAC2HDAC10HDAC6
SCHEMBL29678249 0.71 ALDH1A1 (0.62) KMT2AALDH1A1MAPK1MEN1
SCHEMBL32676372 0.69 MAPT (0.37) KMT2AALDH1A1L3MBTL1MEN1CYP1A2
SCHEMBL3035099 0.68 EGFR (0.41) HDAC1HDAC3KMT2AALDH1A1MAPK1
SCHEMBL29799761 0.67 CYP3A4 (0.39) ALDH1A1MAPK13MAPK12MAPK11MAPK14
SCHEMBL933021 0.67 CYP3A4 (0.39) ALDH1A1MAPK13MAPK12MAPK11MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1608627-A4 BICYCLIC ANILIDE SPIROHYDANTOIN CGRP RECEPTOR ANTAGONISTS MERCK & CO INC (US) 2007-08-01 EP disclosed
EP-1608627-A2 BICYCLIC ANILIDE SPIROHYDANTOIN CGRP RECEPTOR ANTAGONISTS Merck & Co. Inc. (US) 2005-12-28 EP disclosed
WO-2004082605-A2 BICYCLIC ANILIDE SPIROHYDANTOIN CGRP RECEPTOR ANTAGONISTS MERCK & CO. INC. (US) 2004-09-30 WO disclosed