SCHEMBL515177

SCHEMBL515177

NNC(=O)c1cccc([N+](=O)[O-])c1C(=O)NN

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSD P07339 1/20 0.73
ALDH1A1 P00352 2/20 0.53
POLB P06746 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.47
KDM4E B2RXH2 3/20 0.47
TSHR P16473 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
CRHBP P24387 1/20 0.45
CRHR2 Q13324 1/20 0.45
GLA P06280 1/20 0.44
KCNMA1 Q12791 1/20 0.44
GPR35 Q9HC97 1/20 0.44
TP53 P04637 1/20 0.43
MAPT P10636 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30015007 1.00 CTSD (0.73) CTSDALDH1A1POLBCYP1A2CYP3A4
SCHEMBL14321321 0.91 CTSD (0.61) CTSDALDH1A1POLBCYP1A2CYP3A4
SCHEMBL7110523 0.90 CTSD (0.69) CTSDALDH1A1POLBCYP1A2CYP3A4
SCHEMBL16515946 0.85 CTSD (0.61) CTSDALDH1A1POLBCYP1A2CYP3A4
SCHEMBL7539226 0.85 CTSD (0.75) CTSDALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL962966 0.84 CTSD (1.00) CTSDALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL782110 0.83 CTSD (0.73) CTSDALDH1A1POLBCYP1A2CYP3A4
SCHEMBL16146050 0.81 ALDH1A1 (0.50) CTSDALDH1A1POLBCYP1A2CYP3A4
SCHEMBL993341 0.80 CTSD (0.52) CTSDALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL15689544 0.78 CTSD (0.65) CTSDALDH1A1CYP2C9SMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 83 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4073266-B1 METHOD FOR CARRYING OUT AN AMPLIFICATION REACTION IN A MICROFLUIDIC APPARATUS BOSCH GMBH ROBERT (DE) 2026-05-27 EP claimed
US-20230002810-A1 Method for Carrying Out an Amplification Reaction in a Microfluidic Apparatus ROBERT BOSCH GMBH (DE) 2023-01-05 US claimed
US-11511348-B2 Three-dimensional printing HEWLETT-PACKARD DEVELOPMENT COMPANY, L.P. (US) 2022-11-29 US claimed
EP-4073266-A1 METHOD FOR CARRYING OUT AN AMPLIFICATION REACTION IN A MICROFLUIDIC APPARATUS Robert Bosch GmbH (DE) 2022-10-19 EP claimed
US-11398630-B2 Method of generating energy from a hydrazide containing anode fuel, and fuel cell IOWA STATE UNIVERSITY RESEARCH FOUNDATION, INC. (US) 2022-07-26 US claimed
US-20210354196-A1 THREE-DIMENSIONAL PRINTING PERIDOT PRINT LLC 2021-11-18 US claimed
WO-2021116322-A1 METHOD FOR CARRYING OUT AN AMPLIFICATION REACTION IN A MICROFLUIDIC APPARATUS ROBERT BOSCH GMBH (DE) 2021-06-17 WO claimed
US-20210005900-A1 METHOD OF GENERATING ENERGY FROM A HYDRAZIDE CONTAINING ANODE FUEL, AND FUEL CELL IOWA STATE UNIVERSITY RESEARCH FOUNDATION, INC. 2021-01-07 US claimed
EP-3755519-A1 THREE-DIMENSIONAL PRINTING Hewlett-Packard Development Company, L.P. (US) 2020-12-30 EP claimed
WO-2020018131-A1 THREE-DIMENSIONAL PRINTING HEWLETT-PACKARD DEVELOPMENT COMPANY, L.P. (US) 2020-01-23 WO claimed
US-9732043-B2 Process for preparing 5-amino-2,3-dihydrophthalazine-1,4-dione monosodium salt BACH PHARMA, INC. (US) 2017-08-15 US claimed
EP-2393361-B1 PHARMACEUTICAL GRADE PHTHALAZINEDIONES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM BACH PHARMA INC (US) 2016-12-07 EP claimed
US-20160237039-A1 PHARMACEUTICAL GRADE PHTHALAZINEDIONES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Occhiuti & Rohlicek LLP 2016-08-18 US claimed
EP-2393361-A1 PHARMACEUTICAL GRADE PHTHALAZINEDIONES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Bach Pharma, Inc. (US) 2011-12-14 EP claimed
US-20100222584-A1 PHARMACEUTICAL GRADE PHTHALAZINEDIONES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM BACH PHARMA, INC. (US) 2010-09-02 US claimed
WO-2010091257-A1 PHARMACEUTICAL GRADE PHTHALAZINEDIONES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM BACH PHARMA, INC. (US) 2010-08-12 WO claimed
EP-4073266-B1 METHOD FOR CARRYING OUT AN AMPLIFICATION REACTION IN A MICROFLUIDIC APPARATUS BOSCH GMBH ROBERT (DE) 2026-05-27 EP disclosed
EP-4144792-B1 PARTICULATE WATER-ABSORBENT RESIN COMPOSITION, ABSORBENT BODY AND ABSORBENT ARTICLE SUMITOMO SEIKA CHEMICALS (JP) 2025-01-08 EP disclosed
US-4743541-A PURIFICATION OF LUMINOL MAST IMMUNOSYSTEMS, INC. (US) 1988-05-10 US disclosed
EP-0214399-A1 Luminescent substrate preparation and its use in specific binding assays Mast Immunosystems, Inc. (US) 1987-03-18 EP disclosed