SCHEMBL5153683

SCHEMBL5153683

CCCCCNC1(c2ccc(Cl)cc2)CCC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2D O15399 2/20 0.46
GRIN3B O60391 2/20 0.46
GRIA1 P42261 2/20 0.46
GRIA2 P42262 2/20 0.46
GRIA3 P42263 2/20 0.46
GRIA4 P48058 2/20 0.46
GRIN1 Q05586 2/20 0.46
GRIN2A Q12879 2/20 0.46
GRIN2B Q13224 2/20 0.46
GRIN2C Q14957 2/20 0.46
GRIN3A Q8TCU5 2/20 0.46
SMN1; SMN2 Q16637 3/20 0.45
SLC6A4 P31645 8/20 0.40
SLC6A3 Q01959 8/20 0.40
SLC6A2 P23975 5/20 0.40
KDM4E B2RXH2 1/20 0.37
GAA P10253 1/20 0.37
TP53 P04637 1/20 0.36
CYP3A4 P08684 1/20 0.36
ALOX15 P16050 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5310517 0.98 GRIN2D (0.47) GRIN2DGRIN3BGRIA1GRIA2GRIA3
Hydrochloric Acid SCHEMBL5308749 0.94 GRIN2D (0.44) GRIN2DGRIN3BGRIA1GRIA2GRIA3
SCHEMBL5309459 0.81 ALOX15 (0.36) GRIN2DGRIN3BGRIA1GRIA2GRIA3
SCHEMBL28148632 0.80 SLC6A4 (0.53) GRIN2DGRIN3BGRIA1GRIA2GRIA3
SCHEMBL9765029 0.79 GRIN2D (0.70) GRIN2DGRIN3BGRIA1GRIA2GRIA3
SCHEMBL25311978 0.79 GRIN2D (0.49) GRIN2DGRIN3BGRIA1GRIA2GRIA3
SCHEMBL5308917 0.78 CYP3A4 (0.46) GRIN2DGRIN3BGRIA1GRIA2GRIA3
Hydrochloric Acid SCHEMBL5306056 0.78 SLC6A4 (0.48) SLC6A4SLC6A3SLC6A2KCNH2
Hydrochloric Acid SCHEMBL5313074 0.77 CYP3A4 (0.48) GRIN2DGRIN3BGRIA1GRIA2GRIA3
Hydrochloric Acid SCHEMBL5312402 0.76 GRIN2D (0.52) GRIN2DGRIN3BGRIA1GRIA2GRIA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1659154-B Process for the preparation of amine stereoisomers APSINTERM LLC 2012-05-30 CN disclosed
WO-2007041677-A9 SOFT TISSUE IMPLANTS AND DRUG COMBINATION COMPOSITIONS, AND USE THEREOF COMBINATORX INC (US) 2007-05-31 WO disclosed
WO-2007041677-A2 SOFT TISSUE IMPLANTS AND DRUG COMBINATION COMPOSITIONS, AND USE THEREOF COMBINATORX, INCORPORATED (US) 2007-04-12 WO disclosed
EP-1497272-A4 METHOD OF PREPARING AMINE STEREOISOMERS APSINTERM LLC (US) 2007-02-07 EP disclosed
EP-1497272-A2 METHOD OF PREPARING AMINE STEREOISOMERS Apsinterm, LLC. (US) 2005-01-19 EP disclosed
WO-2003091207-A2 METHOD OF PREPARING AMINE STEREOISOMERS APSINTERM, LLC. (US) 2003-11-06 WO disclosed