SCHEMBL5155154

SCHEMBL5155154

O=C1CSC(c2ccccc2Cl)N1CC(Cc1ccccc1)C1=COCO1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.42
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
KMT2A Q03164 4/20 0.38
MEN1 O00255 3/20 0.38
ACHE P22303 2/20 0.38
CACNA1B Q00975 2/20 0.38
POLB P06746 2/20 0.37
NPSR1 Q6W5P4 2/20 0.35
KDM4E B2RXH2 1/20 0.35
HPGD P15428 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5151419 0.84 KMT2A (0.46) ALDH1A1CA1CA2CA9KMT2A
SCHEMBL5156370 0.82 CACNA1B (0.38) ALDH1A1KMT2AMEN1CACNA1BPOLB
SCHEMBL5156718 0.81 MEN1 (0.43) ALDH1A1KMT2AMEN1CACNA1BPOLB
SCHEMBL5149508 0.80 MEN1 (0.44) ALDH1A1KMT2AMEN1ACHEPOLB
SCHEMBL5152312 0.80 HCRTR1 (0.46) ALDH1A1KMT2AMEN1
SCHEMBL5151511 0.80 KMT2A (0.33) ALDH1A1KMT2AMEN1CACNA1BPOLB
SCHEMBL5155501 0.79 MEN1 (0.43) ALDH1A1KMT2AMEN1POLBNPSR1
SCHEMBL6824250 0.78 CACNA1B (0.61) CACNA1B
SCHEMBL5151385 0.78 KMT2A (0.38) ALDH1A1KMT2AMEN1POLBNPSR1
SCHEMBL5156971 0.77 KMT2A (0.37) ALDH1A1KMT2AMEN1CACNA1BPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7223754-B2 Thiazolidinone, oxazolidinone, and imidazolone derivatives for treating lower urinary tract and related disorders DYNOGEN PHARMACEUTICALS, INC. (US) 2007-05-29 US disclosed
US-20070066597-A1 Thiazolidinone, oxazolidinone, and imidazolone derivatives for treating lower urinary tract and related disorders DYNOGEN PHARMACEUTICALS, INC. (US) 2007-03-22 US disclosed
US-20050148587-A1 Thiazolidinone, oxazolidinone, and imidazolone derivatives for treating lower urinary tract and related disorders DYNOGEN PHARMACEUTICALS, INC. (US) 2005-07-07 US disclosed
US-20050113421-A1 Thiazolidinone, oxazolidinone, and imidazolone derivatives for treating non-inflammatory gastrointestinal tract disorders DYNOGEN PHARMACEUTICALS, INC. (US) 2005-05-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050113421-A1 Thiazolidinone, oxazolidinone, and imidazolone derivatives for treating non-inflammatory gastrointestinal tract disorders TRPV2, RYR2, VDAC2 ALDH1A1 3381/4885CA1 3059/4885CA2 171/4885
US-20070066597-A1 Thiazolidinone, oxazolidinone, and imidazolone derivatives for treating lower urinary tract and related disorders RYR2, CACNB2, CACNA1I ALDH1A1 1370/4885CA1 3201/4885CA2 128/4885
US-20050148587-A1 Thiazolidinone, oxazolidinone, and imidazolone derivatives for treating lower urinary tract and related disorders RYR2, CACNB2, CACNA1I ALDH1A1 1370/4885CA1 3201/4885CA2 128/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.