SCHEMBL5155242

SCHEMBL5155242

CCOC(=O)C(N)Cc1ccc(C(N)(CC)CC)cc1

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GRB2 P62993 1/20 0.42
EPHX2 P34913 6/20 0.40
PPARG P37231 3/20 0.40
PTPN1 P18031 2/20 0.40
TPH1 P17752 2/20 0.39
SLC7A5 Q01650 2/20 0.38
MMP8 P22894 1/20 0.38
ALPI P09923 1/20 0.37
PKM P14618 1/20 0.37
PTGS1 P23219 1/20 0.37
XIAP P98170 1/20 0.37
CPB2 Q96IY4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5150701 0.89 GRB2 (0.40) GRB2EPHX2PPARGPTPN1TPH1
SCHEMBL7960935 0.86 SLC7A5 (0.48) GRB2EPHX2PPARGPTPN1TPH1
SCHEMBL5310295 0.85 LMNA (0.46) GRB2EPHX2PPARGPTPN1
SCHEMBL5154257 0.84 GRB2 (0.41) GRB2EPHX2PPARGPTPN1TPH1
SCHEMBL10179224 0.84 PPARG (0.55) GRB2EPHX2PPARGPTPN1
SCHEMBL10181180 0.84 PPARG (0.55) GRB2EPHX2PPARGPTPN1
SCHEMBL20543461 0.81 SLC7A5 (0.44) PPARGTPH1SLC7A5MMP8ALPI
SCHEMBL21117856 0.81 SLC7A5 (0.44) PPARGTPH1SLC7A5MMP8ALPI
SCHEMBL14139328 0.81 SLC7A5 (0.44) PPARGTPH1SLC7A5MMP8ALPI
SCHEMBL9967935 0.81 SLC7A5 (0.44) PPARGTPH1SLC7A5MMP8ALPI

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7157454-B2 Derivatives of n-(arylsulfonyl)beta-aminoacids comprising a substituted aminomethyl group, the preparation method thereof and the pharmaceutical compositions containing same SANOFI-AVENTIS (FR) 2007-01-02 US disclosed
US-20040116353-A1 Derivatives of n-(arylsulfonyl)beta-aminoacids comprising a substituted aminomethyl group, the preparation method thereof and the pharmaceutical compositions containing same SANOFI (FR) 2004-06-17 US disclosed