SCHEMBL5155261

SCHEMBL5155261

CCC(O)NC(CC(N)=O)C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ECE1 P42892 2/20 0.42
ITGB2 P05107 2/20 0.37
ICAM1 P05362 2/20 0.37
ITGAL P20701 2/20 0.37
TGFBR1 P36897 1/20 0.37
CA2 P00918 4/20 0.36
CA1 P00915 3/20 0.36
ALDH1A1 P00352 2/20 0.36
RAB9A P51151 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
PDCD1LG2 Q9BQ51 1/20 0.35
CD274 Q9NZQ7 1/20 0.35
KDM4E B2RXH2 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7605718 0.85 ECE1 (0.41) ECE1ITGB2ICAM1ITGALTGFBR1
SCHEMBL23222804 0.82 ECE1 (0.47) ECE1ITGB2ICAM1ITGALTGFBR1
SCHEMBL20988053 0.82 ECE1 (0.44) ECE1ITGB2ICAM1ITGALTGFBR1
SCHEMBL3364509 0.81 KMT2A (0.42) TGFBR1CA2CA1KMT2A
SCHEMBL5158281 0.81 KMT2A (0.42) TGFBR1CA2CA1KMT2A
SCHEMBL28686537 0.81 GPR84 (0.44) ECE1MAPT
SCHEMBL8601335 0.81 ECE1 (0.47) ECE1ITGB2ICAM1ITGALTGFBR1
SCHEMBL10610009 0.80 ECE1 (0.49) ECE1ITGB2ICAM1ITGALTGFBR1
SCHEMBL5155757 0.80 ECE1 (0.49) ECE1ITGB2ICAM1ITGALTGFBR1
SCHEMBL16750044 0.78 ECE1 (0.50) ECE1ITGB2ICAM1ITGALTGFBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1322411-B1 COLLOIDAL SUSPENSION OF SUBMICRONIC PARTICLES FOR CARRYING ACTIVE PRINCIPLES AND THEIR MODE OF PREPARATION FLAMEL TECH SA (FR) 2007-01-17 EP claimed
EP-1088020-B1 FUNCTIONALISED POLYMERS OF ALPHA-AMINO ACIDS AND THE METHOD OF PREPARATION THEREOF USTAV MAKROMOLEKULARNI CHEMIE (CZ) 2002-12-18 EP claimed
EP-1088020-A1 FUNCTIONALISED POLYMERS OF ALPHA-AMINO ACIDS AND THE METHOD OF PREPARATION THEREOF USTAV MAKROMOLEKULARNI CHEMIE AKADEMIE VED CESKE REPUBLIKY (CZ) 2001-04-04 EP claimed
WO-1999064495-A1 FUNCTIONALISED POLYMERS OF α-AMINO ACIDS AND THE METHOD OF PREPARATION THEREOF ÚSTAV MAKROMOLEKULÁRNÍ CHEMIE AKADEMIE VĚD ČESKÉ REPUBLIKY (CZ) 1999-12-16 WO claimed
EP-1322411-B1 COLLOIDAL SUSPENSION OF SUBMICRONIC PARTICLES FOR CARRYING ACTIVE PRINCIPLES AND THEIR MODE OF PREPARATION FLAMEL TECH SA (FR) 2007-01-17 EP disclosed
EP-1322411-A1 COLLOIDAL SUSPENSION OF SUBMICRONIC PARTICLES FOR CARRYING ACTIVE PRINCIPLES AND THEIR MODE OF PREPARATION FLAMEL TECHNOLOGIES (FR) 2003-07-02 EP disclosed
WO-2002028521-A1 COLLOIDAL SUSPENSION OF SUBMICRONIC PARTICLES FOR CARRYING ACTIVE PRINCIPLES AND THEIR MODE OF PREPARATION FLAMEL TECHNOLOGIES (FR) 2002-04-11 WO disclosed