SCHEMBL5155602

SCHEMBL5155602

NC(=O)c1ccccc1C1=NNC=CC=C1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCAT2 O15382 1/20 0.45
CSNK1A1 P48729 2/20 0.43
DYRK1B Q9Y463 2/20 0.43
TYRO3 Q06418 1/20 0.43
NUDT1 P36639 1/20 0.39
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
KEAP1 Q14145 1/20 0.37
NFE2L2 Q16236 1/20 0.37
KDM4E B2RXH2 2/20 0.37
ALDH1A1 P00352 1/20 0.37
MAPT P10636 1/20 0.37
HPGD P15428 1/20 0.37
TSHR P16473 1/20 0.37
HSD17B10 Q99714 1/20 0.37
CHEK1 O14757 2/20 0.35
METAP2 P50579 1/20 0.35
PARP1 P09874 6/20 0.35
GRM5 P41594 1/20 0.35
ALOX5AP P20292 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29576202 0.86 ALDH1A1 (0.43) NPC1RAB9AKDM4EALDH1A1MAPT
SCHEMBL30514077 0.70 BCAT2 (0.74) BCAT2CSNK1A1DYRK1BTYRO3NUDT1
SCHEMBL210767 0.70 BCAT2 (0.74) BCAT2CSNK1A1DYRK1BTYRO3NUDT1
SCHEMBL7151091 0.70 BCAT2 (0.45) BCAT2CSNK1A1DYRK1BTYRO3NUDT1
SCHEMBL30586908 0.70 BCAT2 (0.45) BCAT2CSNK1A1DYRK1BTYRO3NUDT1
SCHEMBL31012518 0.68 BCAT2 (0.71) BCAT2CSNK1A1DYRK1BTYRO3NUDT1
SCHEMBL1110181 0.68 BCAT2 (0.71) BCAT2CSNK1A1DYRK1BTYRO3NUDT1
Hydrochloric Acid SCHEMBL16463881 0.68 BCAT2 (0.71) BCAT2CSNK1A1DYRK1BTYRO3NUDT1
SCHEMBL3969262 0.68
Hydrochloric Acid SCHEMBL3963502 0.66

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1740185-A1 BENZODIAZEPINES FOR TREATING OR PREVENTING RSV INFECTION Arrow Therapeutics Limited (GB) 2007-01-10 EP disclosed
EP-1727551-A1 PHARMACEUTICAL COMPOSITION COMPRISING A BENZODIAZEPINE DERIVATIVE AND A INHIBITOR OF THE RSV FUSION PROTEIN Arrow Therapeutics Limited (GB) 2006-12-06 EP disclosed
WO-2005089770-A1 BENZODIAZEPINES FOR TREATING OR PREVENTING OR PREVENTING RSV INFECTION ARROW THERAPEUTICS LIMITED (GB) 2005-09-29 WO disclosed
WO-2005090319-A1 PROCESS FOR PREPARING BENZODIAZEPINES ARROW THERAPEUTICS LIMITED (GB) 2005-09-29 WO disclosed
WO-2005089771-A1 PHARMACEUTICAL COMPOSITION COMPRISING A BENZODIAZEPINE DERIVATIVE AND A INHIBITOR OF THE RSV FUSION PROTEIN ARROW THERAPEUTICS LIMITED (GB) 2005-09-29 WO disclosed
US-5795887-A Method of inducing cholecystokinin agonist activity using 1,4- Benzodiazepine compounds GLAXO WELLCOME INC. (US) 1998-08-18 US disclosed