SCHEMBL5156205

SCHEMBL5156205

COc1ccc(Cc2cc(-c3ccncc3)n[nH]2)cc1OC

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.49
KMT2A Q03164 3/20 0.49
CA2 P00918 1/20 0.49
CYP11B1 P15538 1/20 0.45
CYP11B2 P19099 1/20 0.45
CYP17A1 P05093 1/20 0.45
ALDH1A1 P00352 3/20 0.44
GAA P10253 3/20 0.44
POLB P06746 2/20 0.44
MPI P34949 1/20 0.44
APOBEC3G Q9HC16 1/20 0.44
GLA P06280 1/20 0.44
PDE4A P27815 3/20 0.44
PDE4B Q07343 3/20 0.44
PDE4C Q08493 3/20 0.44
PDE4D Q08499 3/20 0.44
CYP3A4 P08684 2/20 0.43
CYP2C9 P11712 2/20 0.43
TSHR P16473 2/20 0.43
CYP2C19 P33261 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5139444 0.90 CYP11B1 (0.46) KDM4EKMT2ACA2CYP11B1CYP11B2
SCHEMBL5109650 0.89 MAPK1 (0.48) KDM4EKMT2ACYP11B1CYP11B2CYP17A1
SCHEMBL5103940 0.89 CYP17A1 (0.48) KDM4EKMT2ACA2CYP11B1CYP11B2
SCHEMBL5100706 0.89 CYP11B1 (0.43) KDM4EKMT2ACYP11B1CYP11B2CYP17A1
SCHEMBL5096786 0.84 COMT (0.58) KDM4EKMT2ACYP11B1CYP11B2CYP17A1
SCHEMBL5111022 0.81 FGFR1 (0.49) KDM4EKMT2ACYP11B1CYP11B2CYP17A1
SCHEMBL5110846 0.80 TACR3 (0.43) CYP11B1CYP11B2CYP17A1PDE4APDE4B
SCHEMBL5096839 0.80 HTR2A (0.39) KDM4EKMT2ACYP11B1CYP11B2CYP17A1
SCHEMBL5104043 0.80 GSK3A (0.46) KDM4EKMT2ACYP17A1ALDH1A1GAA
SCHEMBL14311768 0.79 CYP11B1 (0.57) KDM4ECYP11B1CYP11B2TSHRSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008004100-A2 THERAPEUTIC COMPOUNDS PFIZER PRODUCTS INC. (US) 2008-01-10 WO disclosed