SCHEMBL5156702

SCHEMBL5156702

CCCN(CCC)C(=O)c1ccc(F)c(Br)c1.CCCN(CCC)C(=O)c1ccc(F)c(C(=O)O)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.45
MLYCD O95822 2/20 0.45
TP53 P04637 1/20 0.41
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
LPAR1 Q92633 2/20 0.40
LPAR5 Q9H1C0 2/20 0.40
EGFR P00533 1/20 0.40
ERBB2 P04626 1/20 0.40
HDAC1 Q13547 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
TRPV3 Q8NET8 1/20 0.39
GABRA1 P14867 1/20 0.38
GABRB2 P47870 1/20 0.38
LMNA P02545 1/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3853802 0.92 MLYCD (0.51) HPGDMLYCDTP53LPAR1LPAR5
SCHEMBL3857013 0.91 HPGD (0.53) HPGDMLYCDTP53CYP1A2CYP2D6
SCHEMBL3853804 0.81 TP53 (0.51) HPGDMLYCDTP53LPAR1LPAR5
SCHEMBL3350813 0.77 HPGD (0.43) HPGDMLYCDTP53LPAR1EGFR
SCHEMBL18767254 0.76 HPGD (0.51) HPGDMLYCDTP53EGFRERBB2
SCHEMBL19623314 0.75 HPGD (0.77) HPGDMLYCDTP53NPSR1EGFR
SCHEMBL9300893 0.72 HPGD (0.58) HPGDMLYCDTP53EGFRERBB2
SCHEMBL18767176 0.71 MLYCD (0.50) HPGDMLYCDTP53LPAR1LPAR5
SCHEMBL144208 0.71 ERN1 (0.48) HPGDMEN1KMT2AHTTALDH1A1
SCHEMBL26314066 0.70 MLYCD (0.64) HPGDMLYCDTP53LPAR1LPAR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1740575-A2 PYRROLIDINE DERIVATIVES USEFUL AS BACE INHIBITORS ELI LILLY AND COMPANY (US) 2007-01-10 EP disclosed
WO-2005108358-A2 PYRROLIDINE DERIVATIVES USEFUL AS BACE INHIBITORS ELI LILLY AND COMPANY (US) 2005-11-17 WO disclosed