SCHEMBL5157795

SCHEMBL5157795

CN(C)C1(Cc2cccc(Cl)c2)CCC(NC(=O)CCC(=O)NCCc2ccc(Oc3ccccc3)cc2)CC1.Cc1cccc(CC2(N(C)C)CCC(NC(=O)CCC(=O)NCc3cccc(C)c3C)CC2)c1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.39
EPHX2 P34913 2/20 0.37
LTA4H P09960 1/20 0.37
ALDH1A1 P00352 7/20 0.37
KMT2A Q03164 4/20 0.37
NR3C1 P04150 2/20 0.37
SMN1; SMN2 Q16637 3/20 0.36
RXFP1 Q9HBX9 1/20 0.36
MEN1 O00255 2/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.35
MAPT P10636 2/20 0.34
LMNA P02545 1/20 0.34
TP53 P04637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL206651 0.89 EPHX2 (0.46) HPGDEPHX2LTA4HALDH1A1KMT2A
SCHEMBL206111 0.84 SSTR4 (0.41) ALDH1A1KMT2AMEN1
SCHEMBL206288 0.84 ALDH1A1 (0.50) HPGDEPHX2ALDH1A1KMT2ASMN1; SMN2
SCHEMBL208454 0.83 ALDH1A1 (0.53) HPGDEPHX2ALDH1A1KMT2ASMN1; SMN2
SCHEMBL206578 0.82 ALDH1A1 (0.45) HPGDALDH1A1KMT2ASMN1; SMN2RXFP1
SCHEMBL207315 0.82 ALDH1A1 (0.44) HPGDEPHX2ALDH1A1KMT2AMAPT
SCHEMBL206736 0.82 HPGD (0.48) HPGDEPHX2ALDH1A1KMT2ASMN1; SMN2
SCHEMBL5159686 0.82 NPC1 (0.40) ALDH1A1KMT2ASMN1; SMN2MAPTTP53
SCHEMBL4084112 0.81 HPGD (0.45) HPGDALDH1A1KMT2AMEN1LMNA
SCHEMBL207581 0.81 POLB (0.46) HPGDEPHX2KMT2ARXFP1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007536323-A 2007-12-13 JP claimed
EP-1745010-A1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES Grünenthal GmbH (DE) 2007-01-24 EP claimed
WO-2005110974-A1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES Grünenthal GmbH (DE) 2005-11-24 WO claimed