SCHEMBL5157937

SCHEMBL5157937

O=C(O)Nc1ccccc1.c1ccc(-c2nccnc2-c2ccccc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 3/20 0.55
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
ALDH1A1 P00352 2/20 0.49
LMNA P02545 1/20 0.49
ATR Q13535 1/20 0.47
TAAR1 Q96RJ0 1/20 0.47
SMN1; SMN2 Q16637 5/20 0.47
TP53 P04637 2/20 0.47
EPHX1 P07099 1/20 0.47
TSHR P16473 1/20 0.47
EPHX2 P34913 1/20 0.47
CDK9 P50750 1/20 0.47
CLK4 Q9HAZ1 1/20 0.47
NPC1 O15118 4/20 0.46
RAB9A P51151 4/20 0.46
MAPT P10636 1/20 0.46
HPGD P15428 1/20 0.46
CASP3 P42574 1/20 0.46
SENP8 Q96LD8 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Biphenyl SCHEMBL28335756 0.82 SMN1; SMN2 (0.61) MEN1KMT2AALDH1A1TAAR1SMN1; SMN2
SCHEMBL2192778 0.81 NTRK1 (0.44) CNR1MEN1KMT2ALMNASMN1; SMN2
SCHEMBL30606833 0.81 ATR (0.64) CNR1MEN1KMT2AALDH1A1LMNA
SCHEMBL7634 0.79 EPHX2 (0.70) KMT2AALDH1A1TAAR1SMN1; SMN2TP53
Benzene SCHEMBL28162617 0.79 EPHX2 (0.70) KMT2AALDH1A1TAAR1SMN1; SMN2TP53
Malonic Acid SCHEMBL11758985 0.79 SLC22A12 (0.47) CNR1LMNATSHRPOLBHTT
Iodide SCHEMBL5706290 0.77 EPHX2 (0.67) KMT2AALDH1A1TAAR1SMN1; SMN2TP53
Hydrochloric Acid SCHEMBL9156069 0.77 EPHX2 (0.67) KMT2AALDH1A1TAAR1SMN1; SMN2TP53
Fluoride SCHEMBL10885265 0.77 EPHX2 (0.67) KMT2AALDH1A1TAAR1SMN1; SMN2TP53
Water SCHEMBL9215020 0.77 EPHX2 (0.67) KMT2AALDH1A1TAAR1SMN1; SMN2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1458690-B1 5,6-DIARYL-PYRAZINE-2-AMIDE DERIVATIVES AS CB1 ANTAGONISTS ASTRAZENECA AB (SE) 2007-02-21 EP claimed