SCHEMBL5158280

SCHEMBL5158280

CCCCNc1cc(C(=O)O)cc(N(C)S(C)(=O)=O)n1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 3/20 0.46
BACE1 P56817 11/20 0.45
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
KDM4D Q6B0I6 2/20 0.40
KDM4E B2RXH2 1/20 0.38
USP2 O75604 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CA2 P00918 1/20 0.38
LMNA P02545 1/20 0.38
HPGD P15428 1/20 0.38
TSHR P16473 1/20 0.38
BLM P54132 1/20 0.38
SLC12A2 P55011 1/20 0.38
HIF1A Q16665 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
HSD17B10 Q99714 1/20 0.38
PTGS2 P35354 1/20 0.38
TLR8 Q9NR97 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3860110 0.89 BACE1 (0.45) HCAR3BACE1PTGS2TLR8
SCHEMBL5159403 0.88 BACE1 (0.42) HCAR3BACE1KDM4EALDH1A1LMNA
SCHEMBL4526201 0.80 BACE1 (0.45) BACE1MAPTKDM4DKDM4EALDH1A1
SCHEMBL5158285 0.80 HCAR3 (0.50) HCAR3GAAMAPTKDM4DKDM4E
SCHEMBL3857905 0.79 HCAR3 (0.45) HCAR3BACE1
SCHEMBL3853328 0.79 HCAR3 (0.45) HCAR3BACE1
SCHEMBL3860002 0.78 HCAR3 (0.44) HCAR3BACE1
SCHEMBL3855704 0.78 HCAR3 (0.44) HCAR3BACE1
SCHEMBL7945785 0.78 BACE1 (0.64) BACE1KDM4D
SCHEMBL4531419 0.78 BACE1 (0.64) BACE1KDM4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1740573-A1 AMIDES AS BACE INHIBITORS ELI LILLY AND COMPANY (US) 2007-01-10 EP disclosed
WO-2005108391-A1 AMIDES AS BACE INHIBITORS ELI LILLY AND COMPANY (US) 2005-11-17 WO disclosed