SCHEMBL5160034

SCHEMBL5160034

CN(C)C1(Cc2cccc(Cl)c2)CCC(NC(=O)CCC(=O)NC2CCc3ccccc32)CC1.CN(C)C1(Cc2cccc(Cl)c2)CCC(NC(=O)CCC(=O)NCCc2ccc(Cl)cc2)CC1.CN(C)C1(Cc2cccc(Cl)c2)CCC(NC(=O)CCC(=O)NCCc2ccc(Cl)cc2Cl)CC1.CN(C)C1(Cc2cccc(Cl)c2)CCC(NC(=O)CCC(=O)NCCc2ccccc2Cl)CC1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 3/20 0.40
HPGD P15428 1/20 0.38
ALDH1A1 P00352 4/20 0.37
MAPT P10636 1/20 0.37
P2RX7 Q99572 2/20 0.36
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
EPHX2 P34913 2/20 0.36
PLAAT3 P53816 1/20 0.36
PLAAT5 Q96KN8 1/20 0.36
PLAAT2 Q9NWW9 1/20 0.36
PLAAT4 Q9UL19 1/20 0.36
METAP2 P50579 1/20 0.36
CCR4 P51679 1/20 0.35
LMNA P02545 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4083007 0.87 DHODH (0.45) DHODHHPGDALDH1A1KMT2AMEN1
SCHEMBL208794 0.86 ALDH1A1 (0.44) HPGDALDH1A1KMT2AMEN1EPHX2
SCHEMBL208016 0.86 HPGD (0.48) HPGDALDH1A1MAPTKMT2AEPHX2
SCHEMBL206834 0.85 DHODH (0.48) DHODHHPGDALDH1A1KMT2AMEN1
SCHEMBL206988 0.84 ALDH1A1 (0.51) HPGDALDH1A1MAPTKMT2AMEN1
Hydrochloric Acid SCHEMBL206061 0.83 ALDH1A1 (0.50) HPGDALDH1A1MAPTKMT2AMEN1
SCHEMBL207293 0.81 DHODH (0.48) DHODHALDH1A1KMT2AMEN1LMNA
SCHEMBL208454 0.81 ALDH1A1 (0.53) HPGDALDH1A1MAPTKMT2AMEN1
SCHEMBL205392 0.81 HPGD (0.46) HPGDALDH1A1MAPTKMT2APLAAT3
SCHEMBL205940 0.81 DHODH (0.55) DHODHALDH1A1KMT2AMEN1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007536323-A 2007-12-13 JP claimed
EP-1745010-A1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES Grünenthal GmbH (DE) 2007-01-24 EP claimed
WO-2005110974-A1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES Grünenthal GmbH (DE) 2005-11-24 WO claimed