SCHEMBL5162144

SCHEMBL5162144

Cc1c(-c2ccc(C[C@H](NC(=O)[C@@H]3CCCN3)C(=O)O)cc2)c(=O)n(C)c(=O)n1C

nearest known ligand 0.58

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 14/20 0.58
ITGA4 P13612 14/20 0.58
ITGB7 P26010 14/20 0.58
CTSC P53634 6/20 0.46
CTSK P43235 2/20 0.42
KCNH2 Q12809 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5160248 0.99 ITGB1 (0.57) ITGB1ITGA4ITGB7CTSCCTSK
Hydrochloric Acid SCHEMBL7423666 0.99 ITGB1 (0.57) ITGB1ITGA4ITGB7CTSCCTSK
SCHEMBL27495108 0.80 CTSC (0.44) ITGB1ITGA4ITGB7CTSCCTSK
SCHEMBL7971253 0.77 CTSC (0.58) ITGB1ITGA4CTSCCTSKKCNH2
SCHEMBL5163361 0.77 ITGA4 (0.55) ITGB1ITGA4ITGB7
SCHEMBL6367397 0.77 CTSC (0.56) CTSCCTSKKCNH2
SCHEMBL6367393 0.77 CTSC (0.56) CTSCCTSKKCNH2
SCHEMBL22127884 0.77 CTSC (0.56) CTSCCTSKKCNH2
SCHEMBL21808154 0.77 CTSC (0.68) CTSCCTSKKCNH2
SCHEMBL601567 0.77 CTSC (0.68) CTSCCTSKKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1237878-B1 4-PYRIMIDINYL-N-ACYL-L-PHENYLALANINES HOFFMANN LA ROCHE (CH) 2007-03-21 EP disclosed
EP-1237878-A2 4-PYRIMIDINYL-N-ACYL-L-PHENYLALANINES F. HOFFMANN-LA ROCHE AG (CH) 2002-09-11 EP disclosed
US-6380387-B1 ANTIINFLAMMATORY AGENTS, ANTIASTHMATICS HOFFMANN-LA ROCHE INC. 2002-04-30 US disclosed
WO-2001042225-A2 4-PYRIMIDINYL-N-ACYL-L-PHENYLALANINES F. HOFFMANN-LA ROCHE AG (CH) 2001-06-14 WO disclosed