SCHEMBL5162459

SCHEMBL5162459

c1cncc(-c2ccno2)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 10/20 0.56
ALDH1A1 P00352 5/20 0.56
CYP3A4 P08684 4/20 0.56
CYP1A2 P05177 1/20 0.56
TDO2 P48775 1/20 0.50
NOTUM Q6P988 1/20 0.48
SMN1; SMN2 Q16637 3/20 0.48
HSD17B10 Q99714 3/20 0.48
KDM4E B2RXH2 2/20 0.48
TP53 P04637 2/20 0.48
HPGD P15428 2/20 0.48
MAPT P10636 2/20 0.48
LMNA P02545 1/20 0.48
ALOX15 P16050 1/20 0.48
HTT P42858 1/20 0.48
CYP2E1 P05181 4/20 0.47
CYP2B6 P20813 4/20 0.47
CYP2C19 P33261 4/20 0.47
CYP2D6 P10635 3/20 0.47
CYP2C9 P11712 3/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3618046 0.81 KDM4E (0.63) ALDH1A1CYP3A4CYP1A2SMN1; SMN2HSD17B10
SCHEMBL136631 0.78 NOTUM (0.61) ALDH1A1CYP1A2TDO2NOTUMSMN1; SMN2
SCHEMBL9768763 0.74 NOTUM (0.77) ALDH1A1CYP1A2NOTUMSMN1; SMN2KDM4E
SCHEMBL30238423 0.74 NOTUM (0.63) ALDH1A1CYP1A2NOTUMSMN1; SMN2HSD17B10
SCHEMBL120088 0.74 CYP2A6 (1.00) CYP2A6ALDH1A1CYP3A4CYP1A2SMN1; SMN2
SCHEMBL29419014 0.74 CYP2A6 (1.00) CYP2A6ALDH1A1CYP3A4CYP1A2SMN1; SMN2
SCHEMBL30473120 0.74 CYP2A6 (1.00) CYP2A6ALDH1A1CYP3A4CYP1A2SMN1; SMN2
SCHEMBL11020717 0.73 NOTUM (0.61) ALDH1A1CYP1A2NOTUMSMN1; SMN2KDM4E
SCHEMBL3195754 0.73
SCHEMBL21408748 0.72 NOTUM (0.50) ALDH1A1CYP1A2NOTUMSMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1758896-A1 PYRIDINYL-ISOXAZOLES AND THEIR USE AS HERBICIDES Bayer CropScience GmbH (DE) 2007-03-07 EP disclosed
WO-2005123726-A1 PYRIDINYL-ISOXAZOLES AND THEIR USE AS HERBICIDES BAYER CROPSCIENCE GMBH (DE) 2005-12-29 WO disclosed
US-20050282707-A1 Pyridinylisoxazoles and their use as herbicides BAYER CROPSCIENCE GMBH (DE) 2005-12-22 US disclosed
US-6927228-B2 Biphenyl compounds usefuf in treatment of human and veterinary medicines such as dermatology, cardivovascular diseases, immune diseases or diseases associated with lipid metabolisms, or in cosmetic formulation GALDERMA RESEARCH & DEVELOPMENT, S.N.C. (FR) 2005-08-09 US disclosed
US-20040039038-A1 Biaromatic compound activators of PPARy-type receptors GALDERMA RESEARCH & DEVELOPMENT S.N.C. (FR) 2004-02-26 US disclosed
US-5356912-A 3-(5-isoxazolyl)-1-methyl-1,2,3,6-tetrahydropyridine useful for treating Alzheimer's disease NOVO NORDISK A/S (DK) 1994-10-18 US disclosed
US-5262427-A Cognition activators for Alzheimer*s disease NOVO NORDISK A/S (DK) 1993-11-16 US disclosed
EP-0316718-A2 Azacyclic compounds and their preparation and use NOVO NORDISK A/S (DK) 1989-05-24 EP disclosed
CN-85105299-A The preparation method of cephem compounds 1987-01-07 CN disclosed
EP-0160969-A2 Cephem compounds Takeda Chemical Industries, Ltd. (JP) 1985-11-13 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040039038-A1 Biaromatic compound activators of PPARy-type receptors PPARG, PPARA, PPARD CYP2A6 156/4885ALDH1A1 378/4885CYP3A4 479/4885
US-20050282707-A1 Pyridinylisoxazoles and their use as herbicides PRDX1, CYP4X1, PRDX4 CYP2A6 142/4885ALDH1A1 238/4885CYP3A4 79/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.