SCHEMBL5162574

SCHEMBL5162574

COC(=O)[C@H](Cc1ccc(I)c(C)c1)NC(=O)OCc1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.56
ALOX15 P16050 1/20 0.56
KYNU Q16719 1/20 0.52
CTSL P07711 2/20 0.52
CTSB P07858 2/20 0.52
CTSS P25774 2/20 0.52
CTSK P43235 1/20 0.51
CYP3A4 P08684 3/20 0.51
TSHR P16473 3/20 0.51
MEN1 O00255 1/20 0.51
MAPT P10636 1/20 0.51
KMT2A Q03164 1/20 0.51
CAPN1 P07384 1/20 0.50
TACR1 P25103 2/20 0.49
ATM Q13315 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5162151 0.86 ALDH1A1 (0.56) ALDH1A1ALOX15KYNUCTSLCTSB
SCHEMBL28577401 0.86 ALDH1A1 (0.56) ALDH1A1ALOX15KYNUCTSLCTSB
SCHEMBL28577399 0.86 ALDH1A1 (0.56) ALDH1A1ALOX15KYNUCTSLCTSB
SCHEMBL2402472 0.85 ALDH1A1 (0.57) ALDH1A1ALOX15KYNUCTSLCTSB
SCHEMBL28586890 0.85 ALDH1A1 (0.57) ALDH1A1ALOX15KYNUCTSLCTSB
Hydrochloric Acid SCHEMBL5162142 0.85 ALDH1A1 (0.55) ALDH1A1ALOX15KYNUCTSLCTSB
SCHEMBL5893140 0.85 ALDH1A1 (0.55) ALDH1A1ALOX15KYNUCTSLCTSB
SCHEMBL5887268 0.84 ALDH1A1 (0.65) ALDH1A1ALOX15KYNUCTSLCTSB
SCHEMBL5887270 0.84 ALDH1A1 (0.65) ALDH1A1ALOX15KYNUCTSLCTSB
SCHEMBL7151822 0.84 ALDH1A1 (0.74) ALDH1A1ALOX15KYNUCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1237878-B1 4-PYRIMIDINYL-N-ACYL-L-PHENYLALANINES HOFFMANN LA ROCHE (CH) 2007-03-21 EP disclosed
EP-1237878-A2 4-PYRIMIDINYL-N-ACYL-L-PHENYLALANINES F. HOFFMANN-LA ROCHE AG (CH) 2002-09-11 EP disclosed
US-6380387-B1 ANTIINFLAMMATORY AGENTS, ANTIASTHMATICS HOFFMANN-LA ROCHE INC. 2002-04-30 US disclosed
WO-2001042225-A2 4-PYRIMIDINYL-N-ACYL-L-PHENYLALANINES F. HOFFMANN-LA ROCHE AG (CH) 2001-06-14 WO disclosed