SCHEMBL5164337

SCHEMBL5164337

CC(Oc1cc2c(cc1N)CCCC2)C1CCCCN1

nearest known ligand 0.37

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 9/20 0.37
SLC6A2 P23975 7/20 0.36
SLC6A4 P31645 7/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2035482 0.79 MEN1 (0.41) SLC6A3SLC6A2SLC6A4MEN1KMT2A
SCHEMBL5164769 0.75 HTR2A (0.36) MEN1KMT2A
SCHEMBL6897901 0.75 CYP3A4 (0.41) SLC6A3SLC6A2SLC6A4MEN1KMT2A
SCHEMBL8792376 0.73 MEN1 (0.48) SLC6A3SLC6A2SLC6A4MEN1KMT2A
SCHEMBL11712126 0.72 SLC6A3 (0.40) SLC6A3SLC6A2SLC6A4MEN1KMT2A
SCHEMBL11715216 0.70 NR4A1 (0.44) SLC6A3SLC6A2SLC6A4MEN1KMT2A
SCHEMBL11715498 0.69 SLC6A3 (0.36) SLC6A3SLC6A2SLC6A4
SCHEMBL6701385 0.69 SLC6A3 (0.42) SLC6A3SLC6A2SLC6A4
SCHEMBL8792804 0.68 MEN1 (0.43) SLC6A3SLC6A2SLC6A4MEN1KMT2A
SCHEMBL8587501 0.68 MEN1 (0.43) SLC6A3SLC6A2SLC6A4MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1765808-A1 BISARYLUREA DERIVATIVES USEFUL FOR INHIBITING CHK1 ICOS Corporation (US) 2007-03-28 EP disclosed
WO-2006012308-A1 BISARYLUREA DERIVATIVES USEFUL FOR INHIBITING CHK1 ICOS CORPORATION (US) 2006-02-02 WO disclosed