SCHEMBL5164827

SCHEMBL5164827

COc1cccc(C(C)(C)F)c1OC

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 7/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
TSHR P16473 1/20 0.41
AR P10275 2/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA4 P22748 1/20 0.41
CA7 P43166 1/20 0.41
CA9 Q16790 1/20 0.41
CA14 Q9ULX7 1/20 0.41
RAB9A P51151 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
TP53 P04637 1/20 0.38
CYP3A4 P08684 1/20 0.38
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10451316 0.86 AR (0.49) NFE2L2SMN1; SMN2TSHRARCA12
SCHEMBL29749364 0.86 AR (0.49) NFE2L2SMN1; SMN2TSHRARCA12
SCHEMBL8417921 0.83 SMN1; SMN2 (0.47) NFE2L2SMN1; SMN2CA12CA1CA2
SCHEMBL31438691 0.83 SMN1; SMN2 (0.47) NFE2L2SMN1; SMN2CA12CA1CA2
SCHEMBL1884282 0.80 SMN1; SMN2 (0.44) NFE2L2SMN1; SMN2CA12CA1CA2
SCHEMBL18537139 0.80 SMN1; SMN2 (0.44) NFE2L2SMN1; SMN2TSHRCA12CA1
SCHEMBL20153912 0.77 SMN1; SMN2 (0.46) NFE2L2SMN1; SMN2TSHRCA12CA1
SCHEMBL5706508 0.76 CA1 (0.46) NFE2L2SMN1; SMN2TSHRCA12CA1
SCHEMBL2128908 0.76 SMN1; SMN2 (0.44) NFE2L2SMN1; SMN2TSHRCA12CA1
SCHEMBL11480225 0.76 SMN1; SMN2 (0.44) NFE2L2SMN1; SMN2TSHRCA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1765793-A1 CETP INHIBITORS Merck and Co., Inc. (US) 2007-03-28 EP disclosed
WO-2006014413-A1 CETP INHIBITORS MERCK & CO., INC. (US) 2006-02-09 WO disclosed