SCHEMBL5165263

SCHEMBL5165263

O=C1N=NC(=O)c2[nH]cnc21

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.44
POLB P06746 1/20 0.44
RXFP1 Q9HBX9 1/20 0.44
KDM4E B2RXH2 1/20 0.39
CYP3A4 P08684 1/20 0.39
MAPT P10636 1/20 0.39
ATIC P31939 1/20 0.35
BRD4 O60885 1/20 0.33
MEN1 O00255 1/20 0.32
BLM P54132 1/20 0.32
KMT2A Q03164 1/20 0.32
MAPK14 Q16539 3/20 0.32
MAPK13 O15264 1/20 0.32
RAF1 P04049 1/20 0.32
MAPK9 P45984 1/20 0.32
MAPK12 P53778 1/20 0.32
MAPK11 Q15759 1/20 0.32
IDO1 P14902 3/20 0.31
GDA Q9Y2T3 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13735762 0.72 ALDH1A1 (0.65) ALDH1A1POLBRXFP1KDM4ECYP3A4
SCHEMBL13735766 0.70 ALDH1A1 (0.63) ALDH1A1POLBRXFP1KDM4ECYP3A4
SCHEMBL2775270 0.67 ALDH1A1 (0.44) ALDH1A1POLBRXFP1KDM4ECYP3A4
SCHEMBL18050892 0.67 ALDH1A1 (0.44) ALDH1A1POLBRXFP1KDM4ECYP3A4
SCHEMBL5742205 0.65 ALDH1A1 (0.52) ALDH1A1POLBRXFP1KDM4ECYP3A4
SCHEMBL9708912 0.64 ALDH1A1 (0.55) ALDH1A1POLBRXFP1KDM4ECYP3A4
SCHEMBL414535 0.61 ALDH1A1 (1.00) ALDH1A1POLBRXFP1KDM4ECYP3A4
SCHEMBL5752168 0.60
SCHEMBL5752165 0.60
SCHEMBL158472 0.58 ALDH1A1 (0.32) ALDH1A1POLBRXFP1ATIC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1763530-A1 IMIDAZOPYRIDAZINE DIONES, THE PRODUCTION THEREOF, AND THE USE OF THE SAME AS A MEDICAMENT Boehringer Ingelheim International GmbH (DE) 2007-03-21 EP claimed
WO-2005087774-A1 IMIDAZOPYRIDAZINE DIONES, THE PRODUCTION THEREOF, AND THE USE OF THE SAME AS A MEDICAMENT BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2005-09-22 WO claimed
JP-4235988-A None JP disclosed
EP-1763530-A1 IMIDAZOPYRIDAZINE DIONES, THE PRODUCTION THEREOF, AND THE USE OF THE SAME AS A MEDICAMENT Boehringer Ingelheim International GmbH (DE) 2007-03-21 EP disclosed
WO-2005087774-A1 IMIDAZOPYRIDAZINE DIONES, THE PRODUCTION THEREOF, AND THE USE OF THE SAME AS A MEDICAMENT BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2005-09-22 WO disclosed
JP-H04235988-A IMIDAZOPYRIDAZINEDIODE DERIVATIVE SANKYO CO LTD 1992-08-25 JP disclosed