SCHEMBL5166123

SCHEMBL5166123

CCOP(=O)(Cc1cc(Br)ccc1Cl)OCC

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.39
HPGD P15428 2/20 0.38
TSHR P16473 3/20 0.37
HTR2A P28223 1/20 0.36
SLC6A4 P31645 1/20 0.36
KCNH2 Q12809 1/20 0.36
MAPT P10636 2/20 0.35
ALDH1A1 P00352 3/20 0.34
HTT P42858 3/20 0.34
KMT2A Q03164 3/20 0.34
MEN1 O00255 2/20 0.34
GAA P10253 2/20 0.34
LMNA P02545 1/20 0.34
CYP1A2 P05177 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14731146 0.88 TSHR (0.40) EGFRHPGDTSHRMAPTALDH1A1
SCHEMBL15316683 0.84 TDP1 (0.43) EGFRHPGDTSHRHTR2ASLC6A4
SCHEMBL12798326 0.84 EGFR (0.40) EGFRHPGDTSHRMAPTALDH1A1
SCHEMBL23364293 0.80 KDM4E (0.44) TSHRMAPTALDH1A1HTTKMT2A
SCHEMBL9448834 0.79 EGFR (0.39) EGFRTSHRMAPTALDH1A1HTT
SCHEMBL901666 0.77 HSD17B10 (0.41) EGFRTSHRSLC6A4KCNH2ALDH1A1
SCHEMBL25540658 0.77 CA1 (0.47) TSHRMAPTALDH1A1KMT2AMEN1
SCHEMBL43286 0.75 GABRA1 (0.44) HPGDTSHRHTR2ASLC6A4KCNH2
SCHEMBL29426994 0.75 GABRA1 (0.44) HPGDTSHRHTR2ASLC6A4KCNH2
SCHEMBL18304415 0.75 PYCR1 (0.39) EGFRTSHRMAPTALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7417032-B2 D-xylopyranosyl-phenyl-substituted cycles, medicaments containing such compounds, their use and process for their manufacture BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-08-26 US disclosed
US-7417032-B2 D-xylopyranosyl-phenyl-substituted cycles, medicaments containing such compounds, their use and process for their manufacture BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-08-26 US disclosed
EP-1773800-A1 D-GLUCOPYRANOSYL PHENYL-SUBSTITUTED CYCLENE, MEDICAMENTS CONTAINING THESE COMPOUNDS, THEIR USE, AND METHOD FOR THE PRODUCTION THEREOF Boehringer Ingelheim International GmbH (DE) 2007-04-18 EP disclosed
WO-2006010557-A1 D-GLUCOPYRANOSYL PHENYL-SUBSTITUTED CYCLENE, MEDICAMENTS CONTAINING THESE COMPOUNDS, THEIR USE, AND METHOD FOR THE PRODUCTION THEREOF BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2006-02-02 WO disclosed