SCHEMBL5166307

SCHEMBL5166307

C/C=C/C(=O)N1C(=O)OCC1c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.43
GAA P10253 1/20 0.43
HTT P42858 1/20 0.43
NPC1 O15118 1/20 0.43
LMNA P02545 1/20 0.43
TP53 P04637 1/20 0.43
HPGD P15428 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
RIPK1 Q13546 2/20 0.39
NAAA Q02083 1/20 0.38
IDH1 O75874 6/20 0.37
AVPR1A P37288 1/20 0.36
GLS O94925 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5371801 1.00 ALDH1A1 (0.43) ALDH1A1GAAHTTNPC1LMNA
SCHEMBL28838633 1.00 ALDH1A1 (0.43) ALDH1A1GAAHTTNPC1LMNA
SCHEMBL5371795 1.00 ALDH1A1 (0.43) ALDH1A1GAAHTTNPC1LMNA
SCHEMBL874439 1.00 ALDH1A1 (0.43) ALDH1A1GAAHTTNPC1LMNA
SCHEMBL874440 1.00 ALDH1A1 (0.43) ALDH1A1GAAHTTNPC1LMNA
SCHEMBL23298241 1.00 ALDH1A1 (0.43) ALDH1A1GAAHTTNPC1LMNA
SCHEMBL874438 1.00 ALDH1A1 (0.43) ALDH1A1GAAHTTNPC1LMNA
SCHEMBL6951727 0.85 NPC1 (0.43) ALDH1A1GAAHTTNPC1LMNA
SCHEMBL3117948 0.85 ALDH1A1 (0.43) ALDH1A1GAAHTTNPC1LMNA
SCHEMBL6950966 0.85 NPC1 (0.43) ALDH1A1GAAHTTNPC1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113166173-A Spiro-sulfonamide derivatives as inhibitors of myeloid leukemia 1(MCL-1) protein 普莱鲁德疗法有限公司 2021-07-23 CN disclosed
EP-3181566-A1 IMIDAZOTRIAZINONE COMPOUNDS Ironwood Pharmaceuticals, Inc. (US) 2017-06-21 EP disclosed
EP-1768952-A2 PREPARATION OF BETA-AMINO ACIDS HAVING AFFINITY FOR THE ALPHA-2-DELTA PROTEIN Warner-Lambert Company LLC (US) 2007-04-04 EP disclosed
WO-2006008612-A2 PREPARATION OF BETA-AMINO ACIDS HAVING AFFINITY FOR THE ALPHA-2-DELTA PROTEIN WARNER-LAMBERT COMPANY LLC (US) 2006-01-26 WO disclosed
US-6169181-B1 HUMAN IMMUNODEFICIENCY VIRUS PROTEINASE INHIBITORS PHARMACIA & UPJOHN COMPANY 2001-01-02 US disclosed
US-5852195-A Pyranone compounds useful to treat retroviral infections PHARMACIA & UPJOHN COMPANY (US) 1998-12-22 US disclosed
US-5668164-A Process for synthesis of chiral cis-and trans-3-amino-4 substituted pyrrolidine compounds ABBOTT LABORATORIES (US) 1997-09-16 US disclosed
US-5618949-A Process for synthesis of chiral cis- and trans-3-amino-4-substituted pyrrolidine compounds ABBOTT LABORATORIES (US) 1997-04-08 US disclosed
EP-0758327-A1 PYRANONE COMPOUNDS USEFUL TO TREAT RETROVIRAL INFECTIONS PHARMACIA & UPJOHN COMPANY (US) 1997-02-19 EP disclosed
WO-1995030670-A2 PYRANONE COMPOUNDS USEFUL TO TREAT RETROVIRAL INFECTIONS PHARMACIA & UPJOHN COMPANY (US) 1995-11-16 WO disclosed