SCHEMBL5166486

SCHEMBL5166486

CC(=O)N(c1c(-c2ccc(OC(=O)O)s2)nc2ccccn12)C(C)(C)CC(C)(C)C

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
ALDH1A1 P00352 4/20 0.34
PKM P14618 3/20 0.33
KMT2A Q03164 1/20 0.33
TOP2A P11388 1/20 0.33
KDM4E B2RXH2 1/20 0.33
HPGD P15428 1/20 0.33
HSD17B10 Q99714 1/20 0.33
MAPT P10636 2/20 0.32
GAA P10253 2/20 0.32
TP53 P04637 1/20 0.32
PKLR P30613 1/20 0.32
NTRK1 P04629 2/20 0.32
ADRA1B P35368 1/20 0.31
MAPK1 P28482 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5167941 0.90 PKM (0.39) SMN1; SMN2CYP1A2CYP2C9CYP2C19ALDH1A1
SCHEMBL5164945 0.88 GAA (0.35) ALDH1A1KMT2AKDM4EHPGDHSD17B10
SCHEMBL5166481 0.86 RPS6KB2 (0.38) SMN1; SMN2CYP1A2CYP2C9CYP2C19ALDH1A1
SCHEMBL5164992 0.77 GAA (0.33) SMN1; SMN2ALDH1A1KMT2AKDM4EHPGD
SCHEMBL5167506 0.76 KLK7 (0.40) ALDH1A1PKMKDM4EHPGDHSD17B10
SCHEMBL6750698 0.75 RPS6KB2 (0.42) SMN1; SMN2ALDH1A1PKMKMT2ATOP2A
SCHEMBL5165554 0.74 GAA (0.46) SMN1; SMN2CYP1A2CYP2C9CYP2C19ALDH1A1
SCHEMBL5165905 0.74 PKM (0.38) SMN1; SMN2CYP1A2CYP2C19ALDH1A1PKM
SCHEMBL5164942 0.73 MKNK1 (0.36) CYP2C9CYP2C19ALDH1A1KMT2AKDM4E
SCHEMBL5165500 0.73 KMT2A (0.37) SMN1; SMN2CYP1A2CYP2C9CYP2C19ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1326613-B2 USE OF SUBSTITUTED IMIDAZO 1,2-A|PYRIDINE-, IMIDAZO ¬1,2-A|PYRIMIDINE AND IMIDAZO ¬1,2-A|PYRAZINE-3-YL-AMINE DERIVATIVES FOR PRODUCING NOS-INHIBITING MEDICAMENTS GRUENENTHAL GMBH (DE) 2007-04-18 EP disclosed
EP-1326613-B1 USE OF SUBSTITUTED IMIDAZO 1,2-A]PYRIDINE-, IMIDAZO [1,2-A]PYRIMIDINE AND IMIDAZO [1,2-A]PYRAZINE-3-YL-AMINE DERIVATIVES FOR PRODUCING NOS-INHIBITING MEDICAMENTS GRUENENTHAL GMBH (DE) 2004-06-02 EP disclosed