SCHEMBL5167523

SCHEMBL5167523

C=C(CN(C)Cc1ccc(C(C)(C)C)cc1)c1ccc(C#N)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 2/20 0.51
KIF11 P52732 1/20 0.45
SIGMAR1 Q99720 4/20 0.44
TMEM97 Q5BJF2 2/20 0.44
POLB P06746 1/20 0.44
NSD2 O96028 1/20 0.42
HIF1A Q16665 1/20 0.41
NR1H4 Q96RI1 1/20 0.38
NR1I2 O75469 1/20 0.38
LMNA P02545 1/20 0.38
ADRA2A P08913 1/20 0.38
CYP2D6 P10635 1/20 0.38
ACHE P22303 1/20 0.38
SLC6A2 P23975 1/20 0.38
HTR2A P28223 1/20 0.38
SLC6A4 P31645 1/20 0.38
KCNH2 Q12809 1/20 0.38
PTGES O14684 1/20 0.38
ALOX5 P09917 1/20 0.38
MAOA P21397 5/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5166710 0.89 SIGMAR1 (0.45) EPHX2SIGMAR1TMEM97NR1H4NR1I2
SCHEMBL5169190 0.85 SIGMAR1 (0.40) EPHX2SIGMAR1TMEM97POLBHIF1A
SCHEMBL5167706 0.85 EPHX2 (0.57) EPHX2KIF11SIGMAR1TMEM97POLB
SCHEMBL5167223 0.84 ESRRG (0.49) EPHX2SIGMAR1TMEM97NR1H4NR1I2
SCHEMBL5165638 0.84 NPC1 (0.45) EPHX2SIGMAR1TMEM97NR1H4NR1I2
SCHEMBL5165543 0.82 MAOA (0.50) EPHX2SIGMAR1TMEM97NR1H4NR1I2
SCHEMBL5166068 0.82 NR1H4 (0.51) EPHX2SIGMAR1TMEM97NR1H4PTGES
Hydrochloric Acid SCHEMBL5168719 0.81 MAOA (0.51) EPHX2SIGMAR1TMEM97NR1H4NR1I2
SCHEMBL5169157 0.78 MAOA (0.49) EPHX2SIGMAR1TMEM97NR1H4NR1I2
SCHEMBL5169554 0.78 MAPT (0.48) EPHX2SIGMAR1TMEM97NR1H4LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1561744-B1 AMINE DERIVATIVES, PROCESS FOR PRODUCING THE SAME AND THEIR USE AS ANTIMYCOTIC AGENT POLA CHEM IND INC (JP) 2007-04-18 EP claimed
EP-1561744-A2 AMINE DERIVATIVES, PROCESS FOR PRODUCING THE SAME AND THEIR USE AS ANTIMYCOTIC AGENT POLA CHEMICAL INDUSTRIES INC. (JP) 2005-08-10 EP claimed
US-6329399-B1 Antifungal amine derivatives and processing for producing the same POLA CHEMICAL INDUSTRIES, INC. (JP) 2001-12-11 US claimed
EP-1020426-A1 AMINE DERIVATIVES AND PROCESS FOR PRODUCING THE SAME POLA CHEMICAL INDUSTRIES, INC. (JP) 2000-07-19 EP claimed
EP-1561744-B1 AMINE DERIVATIVES, PROCESS FOR PRODUCING THE SAME AND THEIR USE AS ANTIMYCOTIC AGENT POLA CHEM IND INC (JP) 2007-04-18 EP disclosed
EP-1561744-A2 AMINE DERIVATIVES, PROCESS FOR PRODUCING THE SAME AND THEIR USE AS ANTIMYCOTIC AGENT POLA CHEMICAL INDUSTRIES INC. (JP) 2005-08-10 EP disclosed
US-6329399-B1 Antifungal amine derivatives and processing for producing the same POLA CHEMICAL INDUSTRIES, INC. (JP) 2001-12-11 US disclosed
EP-1020426-A1 AMINE DERIVATIVES AND PROCESS FOR PRODUCING THE SAME POLA CHEMICAL INDUSTRIES, INC. (JP) 2000-07-19 EP disclosed