SCHEMBL5168734

SCHEMBL5168734

Nc1cc(C(F)(F)F)c(-n2cnc(Br)c2)cc1C(=O)O

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CFTR P13569 5/20 0.40
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
HSD17B10 Q99714 1/20 0.38
ASPH Q12797 1/20 0.37
HSP90AA1 P07900 1/20 0.34
GLA P06280 1/20 0.34
AR P10275 1/20 0.33
CA12 O43570 1/20 0.32
CA9 Q16790 1/20 0.32
IDO1 P14902 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5166699 0.86 CFTR (0.52) CFTRKDM4EALDH1A1HPGDHSD17B10
SCHEMBL5167410 0.72 CFTR (0.53) CFTRKDM4EALDH1A1HPGDHSD17B10
SCHEMBL5165199 0.72 CFTR (0.53) CFTRKDM4EALDH1A1HPGDHSD17B10
SCHEMBL21666169 0.72 CFTR (0.51) CFTRKDM4EALDH1A1HPGDHSD17B10
SCHEMBL5165019 0.71 MAPK1 (0.37) CFTRKDM4EALDH1A1
SCHEMBL31356641 0.70 MAP3K5 (0.43) KDM4EASPH
SCHEMBL27381136 0.70 HCAR1 (0.48) ALDH1A1AR
SCHEMBL6602353 0.69 NOTUM (0.35)
SCHEMBL5166472 0.69 CFTR (0.49) CFTRKDM4EALDH1A1HPGDHSD17B10
SCHEMBL5167408 0.68 CFTR (0.60) CFTRKDM4EALDH1A1HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1773788-A2 QUINAZOLINE DERIVATIVES NOVARTIS-PHARMA GMBH (AT) 2007-04-18 EP disclosed
WO-2006010591-A2 QUINAZOLINE DERIVATIVES NOVARTIS AG (CH) 2006-02-02 WO disclosed