SCHEMBL5168924

SCHEMBL5168924

CN(C)C1(c2cccs2)CCC(NC2CCCCCCC2)CC1

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 7/20 0.54
OPRL1 P41146 7/20 0.54
SLC6A4 P31645 1/20 0.41
SLC6A3 Q01959 1/20 0.40
ALDH1A1 P00352 3/20 0.39
HPGD P15428 3/20 0.39
RAB9A P51151 2/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
TSHR P16473 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C19 P33261 1/20 0.39
NPC1 O15118 1/20 0.39
SLC6A2 P23975 1/20 0.39
PRCP P42785 1/20 0.38
SIGMAR1 Q99720 1/20 0.38
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5165622 0.99 OPRM1 (0.52) OPRM1OPRL1SLC6A4SLC6A3ALDH1A1
SCHEMBL3409128 0.81 OPRM1 (0.67) OPRM1OPRL1SLC6A4SLC6A3MEN1
SCHEMBL5166902 0.80 OPRM1 (0.48) OPRM1OPRL1SLC6A4
SCHEMBL5166917 0.80 OPRL1 (0.51) OPRM1OPRL1SLC6A4KMT2ACYP1A2
Hydrochloric Acid SCHEMBL5165321 0.79 OPRM1 (0.47) OPRM1OPRL1
Hydrochloric Acid SCHEMBL5163924 0.79 OPRL1 (0.50) OPRM1OPRL1KMT2ACYP1A2CYP3A4
SCHEMBL20866603 0.78 OPRL1 (0.59) OPRM1OPRL1SLC6A3SLC6A2
SCHEMBL4076511 0.78 OPRL1 (0.59) OPRM1OPRL1SLC6A4SLC6A3SLC6A2
SCHEMBL5164120 0.77 OPRL1 (0.60) OPRM1OPRL1
Hydrochloric Acid SCHEMBL5165769 0.76 OPRL1 (0.61) OPRM1OPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1392641-B1 SUBSTITUTED CYCLOHEXANE-1,4-DIAMINE DERIVATIVES GRUENENTHAL GMBH (DE) 2007-04-11 EP claimed
EP-1385493-A1 SUBSTITUTED CYCLOHEXAN-1,4-DIAMINE DERIVATIVES WITH CONSTIPATING AND PERIPHERAL ANALGESIC PROPERTIES Grünenthal GmbH (DE) 2004-02-04 EP disclosed
WO-2002089783-A1 SUBSTITUTED CYCLOHEXAN-1,4-DIAMINE DERIVATIVES WITH CONSTIPATING AND PERIPHERAL ANALGESIC PROPERTIES Grünenthal GmbH (DE) 2002-11-14 WO disclosed