SCHEMBL5168948

SCHEMBL5168948

COc1ccc(-c2cnc(Nc3ccc(C(=O)CN4CCNCC4)cc3)nc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.49
KDM4E B2RXH2 1/20 0.48
LMNA P02545 1/20 0.48
HDAC3 O15379 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC2 Q92769 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
CCNC P24863 1/20 0.46
CDK8 P49336 1/20 0.46
MKNK2 Q9HBH9 1/20 0.45
IKBKB O14920 1/20 0.44
CHUK O15111 1/20 0.44
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
SYK P43405 1/20 0.43
CSNK2A1 P68400 1/20 0.43
PKM P14618 1/20 0.42
KDR P35968 1/20 0.42
CHEK1 O14757 1/20 0.41
NTRK2 Q16620 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1735187 0.85 CCNC (0.63) HDAC3HDAC1HDAC2HDAC6CCNC
SCHEMBL1735164 0.82 SYK (0.55) IKBKBCHUKSYK
SCHEMBL13605386 0.81 MCHR1 (0.50) IKBKBCHUKSYKESR1
SCHEMBL4873274 0.81 ALDH1A1 (0.71) ALDH1A1KDM4ELMNAMEN1KMT2A
SCHEMBL1734133 0.81 SIGMAR1 (0.50) IKBKBCHUKSYKKDR
Hydrochloric Acid SCHEMBL3844533 0.80 ALDH1A1 (0.69) ALDH1A1KDM4ELMNAMEN1KMT2A
SCHEMBL3643668 0.78 ALDH1A1 (0.45) ALDH1A1MEN1KMT2ACSNK2A1GRM5
SCHEMBL27717813 0.78 HDAC1 (0.63) HDAC3HDAC1HDAC2HDAC6MEN1
SCHEMBL12443599 0.77 CCNC (0.52) HDAC3HDAC1HDAC2HDAC6CCNC
SCHEMBL13605624 0.77 GRM5 (0.65) ALDH1A1KDM4EHDAC3HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1928236-A2 DIARYLAMINE-CONTAINING COMPOUNDS AND COMPOSITIONS, AND THEIR USE AS MODULATORS OF C-KIT RECEPTORS IRM, LLC (BM) 2008-06-11 EP claimed
WO-2007038669-A2 DIARYLAMINE-CONTAINING COMPOUNDS AND COMPOSITIONS, AND THEIR USE AS MODULATORS OF C-KIT RECEPTORS IRM LLC (BM) 2007-04-05 WO claimed