SCHEMBL5169527

SCHEMBL5169527

O=C(O)/C=C/c1cnc(NC2CCN(CCc3ccccc3)C2)c(F)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.44
HTR2A P28223 2/20 0.44
HTR2C P28335 2/20 0.44
HTR2B P41595 2/20 0.44
DRD2 P14416 1/20 0.44
OPRM1 P35372 2/20 0.42
CXCR3 P49682 1/20 0.42
CCR3 P51677 1/20 0.42
HDAC1 Q13547 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
DRD4 P21917 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
GAA P10253 1/20 0.41
TSHR P16473 1/20 0.41
FLT3 P36888 1/20 0.40
TYRO3 Q06418 1/20 0.40
MERTK Q12866 1/20 0.40
GAS6 Q14393 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4225135 1.00 SIGMAR1 (0.44) SIGMAR1HTR2AHTR2CHTR2BDRD2
SCHEMBL4225127 1.00 SIGMAR1 (0.44) SIGMAR1HTR2AHTR2CHTR2BDRD2
SCHEMBL4222248 0.91 SIGMAR1 (0.52) SIGMAR1HTR2AHTR2CHTR2BDRD2
SCHEMBL4222255 0.91 SIGMAR1 (0.52) SIGMAR1HTR2AHTR2CHTR2BDRD2
Hydrochloric Acid SCHEMBL4232002 0.91 HDAC1 (0.50) SIGMAR1HTR2AHTR2CHTR2BDRD2
Hydrochloric Acid SCHEMBL4231998 0.91 HDAC1 (0.50) SIGMAR1HTR2AHTR2CHTR2BDRD2
SCHEMBL4215372 0.87 ROCK2 (0.47) SIGMAR1HTR2AHTR2CHTR2BDRD2
SCHEMBL4215365 0.87 ROCK2 (0.47) SIGMAR1HTR2AHTR2CHTR2BDRD2
SCHEMBL4864890 0.84 SIGMAR1 (0.49) SIGMAR1HTR2AHTR2CHTR2BDRD2
SCHEMBL4864879 0.84 SIGMAR1 (0.49) SIGMAR1HTR2AHTR2CHTR2BDRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1776357-A1 HYDROXYAMIDE COMPOUNDS HAVING ACTIVITY AS INHIBITORS OF HISTONE DEACETYLASE (HDAC) Astellas Pharma Inc. (JP) 2007-04-25 EP disclosed
WO-2006016680-A1 HYDROXYAMIDE COMPOUNDS HAVING ACTIVITY AS INHIBITORS OF HISTONE DEACETYLASE (HDAC) ASTELLAS PHARMA INC. (JP) 2006-02-16 WO disclosed