SCHEMBL5173442

SCHEMBL5173442

N#Cc1cc([N+](=O)[O-])c2sc(OC(N)=O)[n+]([O-])c2c1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 5/20 0.69
MTOR P42345 1/20 0.69
VCAM1 P19320 3/20 0.40
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
GRIN2D O15399 1/20 0.34
GRIN3B O60391 1/20 0.34
GRIN1 Q05586 1/20 0.34
GRIN2A Q12879 1/20 0.34
GRIN2B Q13224 1/20 0.34
GRIN2C Q14957 1/20 0.34
GRIN3A Q8TCU5 1/20 0.34
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32
HPGD P15428 1/20 0.32
CCR6 P51684 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29653627 0.82 PLK1 (1.00) PLK1MTORVCAM1CYP1A2CYP3A4
SCHEMBL5171474 0.82 PLK1 (1.00) PLK1MTORVCAM1CYP1A2CYP3A4
SCHEMBL5169861 0.79 PLK1 (0.69) PLK1MTORCYP1A2CYP3A4CYP2D6
SCHEMBL5171117 0.76 PLK1 (0.71) PLK1MTORCYP1A2CYP3A4CYP2D6
SCHEMBL19192207 0.74 PLK1 (0.71) PLK1MTORVCAM1CYP1A2CYP3A4
SCHEMBL5172975 0.68 PLK1 (0.41) PLK1MTORCYP1A2CYP3A4CYP2D6
SCHEMBL5172960 0.68 PLK1 (0.62) PLK1MTORCYP1A2CYP3A4CYP2D6
SCHEMBL5173246 0.66 PLK1 (0.60) PLK1MTORCYP1A2CYP3A4CYP2D6
SCHEMBL28626079 0.64 VCAM1 (0.59) PLK1MTORVCAM1CYP3A4MAPT
SCHEMBL5173548 0.63 PLK1 (0.71) PLK1MTORCYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1589967-B1 BENZTHIAZOLE-3 OXIDES USEFUL FOR THE TREATMENT OF PROLIFERATIVE DISORDERS CYCLACEL LTD (GB) 2007-05-09 EP claimed