SCHEMBL5175689

SCHEMBL5175689

CCCCNc1nc(N)nc(Cl)c1NC=O

nearest known ligand 0.55

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 19/20 0.55
TLR7 Q9NYK1 8/20 0.50
L3MBTL1 Q9Y468 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13300376 0.82 ALDH1A1 (0.38) TLR8TLR7
SCHEMBL17693700 0.79 TLR8 (0.57) TLR8TLR7
SCHEMBL8695685 0.79 TLR8 (0.64) TLR8TLR7L3MBTL1
SCHEMBL11752787 0.79 TLR8 (0.73) TLR8TLR7L3MBTL1
SCHEMBL17035544 0.78 TLR8 (0.59) TLR8TLR7L3MBTL1
SCHEMBL19495041 0.77 TLR8 (0.71) TLR8TLR7
SCHEMBL13300422 0.77 ALDH1A1 (0.35) TLR8
SCHEMBL20434302 0.76 TLR8 (0.69) TLR8TLR7L3MBTL1
SCHEMBL2848341 0.75 TLR8 (0.52) TLR8TLR7
SCHEMBL536664 0.74 CHUK (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0684236-B2 Process of preparation of N-(2-Amino-4,6-dichloropyrimidin-5-yl)formamide LONZA AG (CH) 2007-12-26 EP disclosed
CN-1193991-C Method for preparing 2,5-diamino-4,6-dichloropyrimidine LONZE AG (CH) 2005-03-23 CN disclosed
CN-1065862-C N- (2-amino-4, 6-dichloropyrimidin-5-yl) formamide and preparation method thereof LONZA AG (CH) 2001-05-16 CN disclosed
CN-1259517-A Method for preparing 2,5-diamino-4,6-dichloropyrimidine LONZE AG (CH) 2000-07-12 CN disclosed
EP-0684236-B1 N-(2-Amino-4,6-dichloropyrimidin-5-yl)formamide and process for its production LONZA AG (CH) 1998-06-24 EP disclosed
US-5744601-A N-(2-amino-4, 6-dichlopyrimidine-5-yl) formanide, and a process for its preparation LONZA AG (CH) 1998-04-28 US disclosed
US-5693800-A N-(2-amino-4,6-dichloropyrimidine-5-yl) formamide and a process for its preparation LONZA AG (CH) 1997-12-02 US disclosed
US-5663340-A N-(2-amino-4,6-dichloropyrimidine-5-yl)formamide, and a process for its preparation LONZA AG (CH) 1997-09-02 US disclosed
US-5583226-A 4,6-dichloropyrimidine and related compounds LONZA AG (CH) 1996-12-10 US disclosed
EP-0684236-A2 N-(2-Amino-4,6-dichloropyrimidin-5-yl)formamide and process for its production LONZA AG (CH) 1995-11-29 EP disclosed