SCHEMBL5176291

SCHEMBL5176291

CN1CCN(c2ccc(-c3nc(N)cc(N)n3)cc2)CC1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.56
MAPT P10636 3/20 0.56
GAA P10253 2/20 0.56
PTK2B Q14289 2/20 0.56
ALDH1A1 P00352 1/20 0.56
ADRA2C P18825 1/20 0.56
GFER P55789 1/20 0.56
KMT2A Q03164 1/20 0.56
ESR2 Q92731 1/20 0.56
HRH4 Q9H3N8 11/20 0.51
JAK2 O60674 1/20 0.51
HRH3 Q9Y5N1 3/20 0.50
HTR6 P50406 1/20 0.50
CHEK1 O14757 2/20 0.49
MAPK1 P28482 1/20 0.49
HTT P42858 1/20 0.49
RECQL P46063 1/20 0.49
FYN P06241 1/20 0.48
NPC1 O15118 1/20 0.48
XBP1 P17861 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1493708 0.77 HTR6 (0.54) KDM4EMAPTGAAPTK2BALDH1A1
SCHEMBL25894824 0.75 MAPT (0.88) KDM4EMAPTGAAPTK2BALDH1A1
SCHEMBL16965450 0.75 JAK2 (0.56) KDM4EMAPTGAAPTK2BALDH1A1
SCHEMBL12892361 0.75 KDM4E (0.55) KDM4EMAPTGAAPTK2BALDH1A1
SCHEMBL28051294 0.74 RPS6KA3 (0.59) KDM4EMAPTGAAPTK2BALDH1A1
SCHEMBL28577095 0.74 MELK (0.65) KDM4EMAPTGAAPTK2BALDH1A1
SCHEMBL14851170 0.74 KDM4E (0.51) KDM4EMAPTGAAPTK2BALDH1A1
SCHEMBL1493668 0.74 HRH4 (0.52) HRH4HRH3
SCHEMBL31173630 0.73 MAPT (0.60) KDM4EMAPTGAAPTK2BALDH1A1
SCHEMBL20475482 0.73 MAPT (0.60) KDM4EMAPTGAAPTK2BALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103121973-A Pyrimidine urea derivatives as kinase inhibitors NOVARTIS AG 2013-05-29 CN disclosed
CN-103121972-A Pyrimidine urea derivatives as kinase inhibitors NOVARTIS AG 2013-05-29 CN disclosed
EP-1761505-A1 PYRIMIDINE UREA DERIVATIVES AS KINASE INHIBITORS Novartis AG (CH) 2007-03-14 EP disclosed
WO-2006000420-A1 PYRIMIDINE UREA DERIVATIVES AS KINASE INHIBITORS NOVARTIS AG (CH) 2006-01-05 WO disclosed