SCHEMBL5178131

SCHEMBL5178131

CCOC(=O)c1ccc2cc(OCCCC3CCCNC3)ccc2n1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ACP1 P24666 5/20 0.46
HRH3 Q9Y5N1 2/20 0.43
MAOA P21397 2/20 0.42
BCHE P06276 1/20 0.42
ACHE P22303 1/20 0.42
MAOB P27338 1/20 0.42
SCN9A Q15858 1/20 0.39
P2RY12 Q9H244 4/20 0.39
PDE3B Q13370 3/20 0.39
PDE3A Q14432 3/20 0.39
PDE2A O00408 2/20 0.39
MAP2K1 Q02750 1/20 0.39
CHEK2 O96017 1/20 0.39
NPY1R P25929 1/20 0.38
EP300 Q09472 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2208858 0.88 HRH3 (0.44) ACP1HRH3SCN9AMAP2K1CHEK2
SCHEMBL1381216 0.83 HRH3 (0.61) ACP1HRH3SCN9A
SCHEMBL1377869 0.83 HRH3 (0.61) HRH3SCN9A
SCHEMBL5178917 0.83 HRH3 (0.51) HRH3SCN9A
SCHEMBL1380830 0.82 HRH3 (0.67) HRH3SCN9A
SCHEMBL1380750 0.81 HRH3 (0.50) HRH3SCN9A
SCHEMBL1381575 0.81 HRH3 (0.56) HRH3SCN9A
SCHEMBL1381719 0.81 HRH3 (0.51) HRH3SCN9A
SCHEMBL1380359 0.80 HRH3 (0.53) ACP1HRH3SCN9AP2RY12PDE3B
SCHEMBL1378414 0.80 SCN9A (0.53) HRH3SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1805166-A1 QUINOLINE DERIVATIVES F. Hoffmann-Roche AG (CH) 2007-07-11 EP disclosed
WO-2006045416-A1 QUINOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2006-05-04 WO disclosed