SCHEMBL5178798

SCHEMBL5178798

COc1c(N2CCN(CCOCCO)CC2)c(F)cc2c(=O)c(OC(=O)NCc3ccc(Cl)cc3C)cn(C3CC3)c12

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 9/20 0.42
ALDH1A1 P00352 4/20 0.42
TDP1 Q9NUW8 3/20 0.42
LMNA P02545 2/20 0.42
POLB P06746 2/20 0.42
NPSR1 Q6W5P4 1/20 0.42
KCNH2 Q12809 3/20 0.41
HPGD P15428 4/20 0.40
HSD17B10 Q99714 2/20 0.40
PRKD3 O94806 1/20 0.40
ALOX15 P16050 1/20 0.40
OPRM1 P35372 1/20 0.40
CLK2 P49760 1/20 0.40
CLK4 Q9HAZ1 1/20 0.40
CYP2C19 P33261 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.38
ATM Q13315 1/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5284805 0.93 ALDH1A1 (0.39) KDM4EALDH1A1TDP1LMNAPOLB
SCHEMBL965915 0.91 KDM4E (0.46) KDM4EALDH1A1TDP1LMNAPOLB
SCHEMBL5278268 0.87 EPHX2 (0.36) KDM4EALDH1A1TDP1LMNAPOLB
SCHEMBL5178320 0.87 KDM4E (0.36) KDM4EALDH1A1TDP1LMNAPOLB
SCHEMBL5282397 0.86 ALDH1A1 (0.40) ALDH1A1POLBOPRM1
SCHEMBL12917365 0.85 KDM4E (0.48) KDM4EALDH1A1TDP1LMNAPOLB
SCHEMBL967809 0.84 ALDH1A1 (0.43) KDM4EALDH1A1TDP1LMNAPOLB
SCHEMBL5181324 0.83 KCNH2 (0.52) KDM4EALDH1A1TDP1LMNAPOLB
SCHEMBL5280454 0.79 EPHX2 (0.36) ALDH1A1POLBOPRM1
SCHEMBL5280465 0.79 EPHX2 (0.36) ALDH1A1POLBOPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1768973-A1 SUBSTITUTED QUINOLONES AiCuris GmbH & Co. KG (DE) 2007-04-04 EP disclosed
WO-2006008046-A1 SUBSTITUTED QUINOLONES AICURIS GMBH & CO. KG (DE) 2006-01-26 WO disclosed