SCHEMBL5284805

SCHEMBL5284805

Cc1cc(Cl)ccc1CNC(=O)Oc1cn(C2CC2)c2c(Cl)c(N3CCN(CCOCCO)CC3)c(F)cc2c1=O

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.39
POLB P06746 2/20 0.39
CHRM2 P08172 1/20 0.39
CHRM1 P11229 1/20 0.39
OPRM1 P35372 1/20 0.39
OPRD1 P41143 1/20 0.39
P2RX7 Q99572 2/20 0.35
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
HTR2A P28223 1/20 0.34
HTR2B P41595 1/20 0.34
KCNH2 Q12809 1/20 0.34
BCL2A1 Q16548 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5282397 0.93 ALDH1A1 (0.40) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL5178798 0.93 KDM4E (0.42) ALDH1A1POLBOPRM1KDM4ELMNA
SCHEMBL967809 0.91 ALDH1A1 (0.43) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL5280465 0.86 EPHX2 (0.36) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL5280454 0.86 EPHX2 (0.36) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL5279342 0.86 EPHX2 (0.36) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL5178320 0.85 KDM4E (0.36) ALDH1A1POLBOPRM1P2RX7KDM4E
SCHEMBL5274263 0.85 ALDH1A1 (0.40) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL966775 0.84 ALDH1A1 (0.44) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL965915 0.84 KDM4E (0.46) ALDH1A1POLBOPRM1KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1768973-B1 SUBSTITUTED QUINOLONES AICURIS GMBH & CO KG (DE) 2007-12-05 EP disclosed