SCHEMBL5178994

SCHEMBL5178994

CCOC(=O)c1cnc(N(C)c2cc(C(C)(C)C)cc(C(C)(C)C)c2)nc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 2/20 0.40
CYP2C19 P33261 2/20 0.40
TDP1 Q9NUW8 1/20 0.40
MAPT P10636 2/20 0.39
MEN1 O00255 1/20 0.39
NPC1 O15118 1/20 0.39
GAA P10253 1/20 0.39
RAB9A P51151 1/20 0.39
KMT2A Q03164 1/20 0.39
MAOB P27338 3/20 0.39
CA12 O43570 3/20 0.39
CA1 P00915 3/20 0.39
CA2 P00918 3/20 0.39
CA7 P43166 3/20 0.39
CA9 Q16790 3/20 0.39
CA14 Q9ULX7 3/20 0.39
P2RY12 Q9H244 1/20 0.39
HDAC3 O15379 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5180005 0.87 RXRA (0.39) CYP2C9CYP2C19TDP1MAPTMEN1
SCHEMBL5178219 0.85 RXRA (0.37) CYP2C9CYP2C19TDP1MAPTMEN1
SCHEMBL5180399 0.81 RXRA (0.44) CYP2C9CYP2C19TDP1MAPTMEN1
SCHEMBL5179646 0.80 KDM4E (0.54) TDP1MAPTMEN1KMT2AHDAC3
SCHEMBL11530672 0.77 ALDH1A1 (0.56) CYP2C9CYP2C19MAPTNPC1GAA
SCHEMBL5665632 0.76 CA12 (0.58) CYP2C9CYP2C19TDP1NPC1CA12
SCHEMBL5179272 0.76 HDAC3 (0.47) CYP2C9CYP2C19TDP1MAPTMEN1
SCHEMBL22235630 0.75 RXRA (0.40) CYP2C19TDP1RAB9ACA1CA2
SCHEMBL3564942 0.74 CYP2C9 (0.47) CYP2C9CYP2C19MAPTMEN1NPC1
SCHEMBL16418625 0.73 CA12 (0.58) CYP2C9CYP2C19TDP1MEN1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1180520-B1 PYRIMIDINE CARBOXYLIC ACID DERIVATIVES INST MED MOLECULAR DESIGN INC (JP) 2007-06-20 EP disclosed
US-6869959-B1 Heterocyclic carboxylic acid derivatives INSTITUTE OF MEDICINAL MOLECULAR DESIGN INC. (JP) 2005-03-22 US disclosed
EP-1180520-A1 HETEROCYCLIC CARBOXYLIC ACID DERIVATIVES Institute of Medicinal Molecular Design, Inc. (JP) 2002-02-20 EP disclosed