SCHEMBL5184705

SCHEMBL5184705

NC(=O)c1ccccc1CC[CH]C(=O)Nc1ccc2ncccc2c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 7/20 0.51
POLB P06746 2/20 0.51
MEN1 O00255 1/20 0.51
MAPT P10636 1/20 0.51
KMT2A Q03164 1/20 0.51
RAB9A P51151 6/20 0.51
ALDH1A1 P00352 2/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
TSHR P16473 1/20 0.50
HSD17B10 Q99714 1/20 0.50
PABPC1 P11940 1/20 0.49
HTT P42858 1/20 0.47
NOTUM Q6P988 1/20 0.45
NAMPT P43490 3/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
SYK P43405 2/20 0.43
CASP3 P42574 1/20 0.43
SENP8 Q96LD8 1/20 0.43
SENP7 Q9BQF6 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5184088 0.92 TRPV1 (0.45) NPC1POLBMEN1MAPTKMT2A
SCHEMBL5185052 0.88 KDM4E (0.48) NPC1POLBMEN1MAPTKMT2A
SCHEMBL5184813 0.87 NPSR1 (0.49) NPC1POLBMAPTRAB9AALDH1A1
SCHEMBL5231291 0.82 PABPC1 (0.58) NPC1POLBMEN1MAPTKMT2A
SCHEMBL4950035 0.82 KDR (0.43) NPC1POLBMAPTRAB9AALDH1A1
SCHEMBL4950199 0.82 KDR (0.39) POLBMAPTRAB9AALDH1A1TSHR
SCHEMBL4950537 0.80 PDE4B (0.43) NPC1MEN1KMT2ARAB9ASMN1; SMN2
SCHEMBL4952020 0.79 CNR1 (0.41) SYKHDAC4
SCHEMBL5185017 0.78 RAB9A (0.46) NPC1POLBMAPTRAB9AALDH1A1
SCHEMBL5185045 0.78 NPC1 (0.49) NPC1POLBMEN1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1758920-A1 BACTERIAL EFFLUX PUMP INHIBITORS AND METHODS OF TREATING BACTERIAL INFECTIONS MPEX PHARMACEUTICALS, INC. (US) 2007-03-07 EP disclosed
WO-2005113579-A1 BACTERIAL EFFLUX PUMP INHIBITORS AND METHODS OF TREATING BACTERIAL INFECTIONS MPEX PHARMACEUTICALS, INC. (US) 2005-12-01 WO disclosed