SCHEMBL5185239

SCHEMBL5185239

O=C(O)[C@@H]1CCCCN1S(=O)(=O)c1ccccc1C(F)(F)F

nearest known ligand 0.61

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 1/20 0.61
HTT P42858 2/20 0.55
KMT2A Q03164 3/20 0.54
MEN1 O00255 1/20 0.54
KCNQ1 P51787 1/20 0.52
ALDH1A1 P00352 3/20 0.50
GAA P10253 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.48
CHRM4 P08173 1/20 0.46
MMP8 P22894 1/20 0.44
MMP12 P39900 1/20 0.44
MMP13 P45452 1/20 0.44
POLB P06746 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3728863 0.96 HCRTR1 (0.65) HCRTR1HTTKMT2AMEN1KCNQ1
SCHEMBL8911492 0.84 HCRTR1 (0.55) HCRTR1HTTALDH1A1GAAMMP8
SCHEMBL8911495 0.84 HCRTR1 (0.55) HCRTR1HTTALDH1A1GAAMMP8
SCHEMBL3441808 0.83 HCRTR1 (0.58) HCRTR1KMT2AMEN1KCNQ1ALDH1A1
SCHEMBL4344983 0.83 HCRTR1 (0.52) HCRTR1KMT2AMEN1KCNQ1ALDH1A1
SCHEMBL3446571 0.83 HCRTR1 (0.57) HCRTR1KMT2AMEN1KCNQ1ALDH1A1
SCHEMBL29783823 0.82 CHRM4 (0.58) HCRTR1KMT2AMEN1KCNQ1L3MBTL1
SCHEMBL3441729 0.81 OPRM1 (0.54) HCRTR1KMT2AMEN1KCNQ1ALDH1A1
SCHEMBL4436227 0.81 OPRM1 (0.54) HCRTR1KMT2AMEN1KCNQ1ALDH1A1
SCHEMBL5173968 0.80 HTT (0.58) HTTALDH1A1MMP8MMP12MMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1778637-A2 FKBP BINDING COMPOSITION AND PHARMACEUTICAL USE THEREOF Aventis Pharmaceuticals, Inc. (US) 2007-05-02 EP disclosed
WO-2006012256-A2 FKBP BINDING COMPOSITION AND PHARMACEUTICAL USE THEREOF AVENTIS PHARMACEUTICALS INC. (US) 2006-02-02 WO disclosed