SCHEMBL5186159

SCHEMBL5186159

COc1ccc(-c2c(C(=O)O)n(CCN3CCOCC3)c3cc(OC)c(OC)cc23)cc1

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 8/20 0.52
EDNRB P24530 5/20 0.52
CNR1 P21554 2/20 0.50
ALDH1A1 P00352 1/20 0.50
TP53 P04637 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
TSHR P16473 1/20 0.50
CNR2 P34972 1/20 0.50
RECQL P46063 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
MAPK1 P28482 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
LMNA P02545 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4591982 0.91 ALDH1A1 (0.49) CNR1ALDH1A1TP53CYP1A2CYP3A4
SCHEMBL5424965 0.91 EDNRA (0.50) EDNRAEDNRB
Hydrochloric Acid SCHEMBL4591984 0.90 ALDH1A1 (0.48) CNR1ALDH1A1TP53CYP1A2CYP3A4
SCHEMBL4592011 0.85 EDNRB (0.52) EDNRAEDNRBALDH1A1LMNA
SCHEMBL4591054 0.85 EDNRA (0.52) EDNRAEDNRB
SCHEMBL4591109 0.82 ALDH1A1 (0.45) EDNRAEDNRBALDH1A1TSHR
SCHEMBL4592550 0.82 KMT2A (0.50) EDNRAEDNRBALDH1A1TDP1
SCHEMBL13990308 0.82 CREBBP (0.47) CNR1ALDH1A1TP53CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL4591112 0.82 ESR1 (0.45) ALDH1A1TSHRLMNA
SCHEMBL4883674 0.82 ALDH1A1 (0.42) EDNRAEDNRBALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1750687-A2 INDOLE AND AZAINDOLE DERIVATIVES WITH ANTITUMOR ACTION NIKEM RESEARCH S.R.L. (IT) 2007-02-14 EP claimed
WO-2005105213-A2 INDOLE AND AZAINDOLE DERIVATIVES WITH ANTITUMOR ACTION NIKEM RESEARCH S.R.L. (IT) 2005-11-10 WO claimed