SCHEMBL5190158

SCHEMBL5190158

COC(=O)N1CCNCC1CC(N)=O

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.36
TSHR P16473 1/20 0.36
CHRNB2 P17787 2/20 0.36
CHRNA4 P43681 2/20 0.36
CHRNB4 P30926 1/20 0.36
CHRNA3 P32297 1/20 0.36
CA1 P00915 4/20 0.34
CA2 P00918 4/20 0.34
CA4 P22748 4/20 0.34
CA9 Q16790 4/20 0.34
CHRNA7 P36544 2/20 0.34
KCNH2 Q12809 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4332678 0.83 TSHR (0.39) PARP1TSHRCHRNB2CHRNA4CHRNB4
SCHEMBL5195457 0.82 FHIT (0.34) PARP1CA1CA2CA4CA9
Hydrochloric Acid SCHEMBL17560393 0.81 TSHR (0.38) PARP1TSHRCHRNB2CHRNA4CHRNB4
SCHEMBL5193793 0.81 GBA2 (0.39) PARP1CA1CA2CA4CA9
SCHEMBL5195326 0.77 LMNA (0.39) CHRNB2CHRNA4CHRNB4CHRNA3CA1
SCHEMBL2919209 0.76 TSHR (0.36) TSHRCA1CA2CA4CA9
SCHEMBL1149942 0.74 PARP1 (0.50) PARP1
SCHEMBL9098808 0.74 PARP1 (0.50) PARP1
SCHEMBL18706103 0.74 LMNA (0.39) CHRNA7KCNH2
SCHEMBL4340453 0.74 TSHR (0.52) TSHRCHRNB2CHRNA4CHRNB4CHRNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0968206-B8 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX INC (US) 2007-01-24 EP disclosed
EP-0968206-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 2000-01-05 EP disclosed
WO-1998037079-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 1998-08-27 WO disclosed