SCHEMBL5190762

SCHEMBL5190762

CC(=O)N1CCN(C(C)c2ccc(Cl)cc2)C(CC(N)=O)C1

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.39
HPGD P15428 1/20 0.39
SLC6A9 P48067 3/20 0.39
CYP3A4 P08684 1/20 0.38
CYP3A5 P20815 1/20 0.38
GPX4 P36969 2/20 0.36
DPP4 P27487 1/20 0.35
DPP7 Q9UHL4 1/20 0.35
HSD11B1 P28845 1/20 0.35
POLB P06746 1/20 0.35
FFAR2 O15552 1/20 0.35
OPRK1 P41145 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5193306 0.88 POLB (0.48) SLC6A9CYP3A4GPX4POLB
SCHEMBL5193461 0.82 HIF1A (0.40) ALDH1A1POLB
SCHEMBL5194017 0.75 ALDH1A1 (0.41) ALDH1A1HPGDCYP3A4POLB
SCHEMBL5193553 0.69 PDGFRB (0.45)
SCHEMBL5193932 0.68 TSHR (0.43) ALDH1A1HSD11B1
SCHEMBL11623725 0.68 CYP3A4 (0.53) ALDH1A1HPGDCYP3A4CYP3A5GPX4
SCHEMBL5192435 0.68 MCHR1 (0.44) ALDH1A1POLBOPRK1
SCHEMBL5213600 0.68 ALDH1A1 (0.51) ALDH1A1POLB
SCHEMBL10266852 0.68 ALDH1A1 (0.48) ALDH1A1HPGDSLC6A9CYP3A4CYP3A5
SCHEMBL2738699 0.68 ALDH1A1 (0.48) ALDH1A1HPGDSLC6A9CYP3A4CYP3A5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0968206-B8 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX INC (US) 2007-01-24 EP disclosed
EP-0968206-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 2000-01-05 EP disclosed
WO-1998037079-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 1998-08-27 WO disclosed