SCHEMBL5192029

SCHEMBL5192029

COc1cccc(CNC(=O)CC2CNCCN2)c1

nearest known ligand 0.57

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.56
HTT P42858 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
POLB P06746 1/20 0.52
HPGD P15428 1/20 0.52
EPHX2 P34913 2/20 0.51
MMP13 P45452 1/20 0.50
KDM4E B2RXH2 1/20 0.48
APEX1 P27695 1/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
NPC1 O15118 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5190305 0.86 ALDH1A1 (0.54) ALDH1A1SMN1; SMN2POLBMEN1KMT2A
SCHEMBL5190550 0.83 ALDH1A1 (0.53) ALDH1A1SMN1; SMN2POLBEPHX2KDM4E
SCHEMBL21162505 0.82 MC4R (0.52) ALDH1A1SMN1; SMN2POLBMEN1KMT2A
SCHEMBL5190702 0.81 GAA (0.49) ALDH1A1KDM4EMEN1KMT2A
SCHEMBL6170662 0.78 HTT (0.67) ALDH1A1HTTSMN1; SMN2POLBHPGD
SCHEMBL17101 0.78 EED (0.61) ALDH1A1
SCHEMBL2250418 0.78 EED (0.61) ALDH1A1
SCHEMBL5193058 0.77 KMT2A (0.45) ALDH1A1SMN1; SMN2HPGDMEN1KMT2A
SCHEMBL5557978 0.76 EED (0.52)
SCHEMBL5557983 0.76 EED (0.52)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0968206-B8 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX INC (US) 2007-01-24 EP claimed
EP-0968206-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 2000-01-05 EP claimed
WO-1998037079-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 1998-08-27 WO claimed