SCHEMBL5193849

SCHEMBL5193849

COc1cccc(CCN2CCCCC2CC(N)=O)c1

nearest known ligand 0.60

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 4/20 0.60
SIGMAR1 Q99720 3/20 0.50
TDP1 Q9NUW8 1/20 0.48
HCRTR1 O43613 1/20 0.47
HCRTR2 O43614 1/20 0.47
DRD2 P14416 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26024360 0.89 HRH3 (0.60) HRH3SIGMAR1TDP1HCRTR1HCRTR2
SCHEMBL5195350 0.86 HRH3 (0.56) HRH3SIGMAR1DRD2
SCHEMBL6802071 0.85 HRH3 (0.66) HRH3SIGMAR1TDP1
SCHEMBL6802079 0.85 HRH3 (0.66) HRH3SIGMAR1TDP1
SCHEMBL5191198 0.84 MAPK1 (0.56) SIGMAR1TDP1HCRTR1HCRTR2DRD2
SCHEMBL8938433 0.80 HRH3 (0.69) HRH3SIGMAR1TDP1
SCHEMBL9752686 0.78 HRH3 (0.69) HRH3SIGMAR1
SCHEMBL5195704 0.77 SPHK2 (0.52) SIGMAR1
SCHEMBL26024361 0.76 TDP1 (0.51) HRH3SIGMAR1TDP1
SCHEMBL5193949 0.76 OPRD1 (0.45) HRH3SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0968206-B8 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX INC (US) 2007-01-24 EP claimed
EP-0968206-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 2000-01-05 EP claimed
WO-1998037079-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 1998-08-27 WO claimed