SCHEMBL5194004

SCHEMBL5194004

CCCn1cc2c(n1)c(N)nc1cccc(C)c12

nearest known ligand 0.58

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 5/20 0.58
TLR7 Q9NYK1 3/20 0.58
ADORA3 P0DMS8 8/20 0.44
ADORA2A P29274 8/20 0.44
ADORA1 P30542 7/20 0.40
ADORA2B P29275 2/20 0.40
PIK3CD O00329 1/20 0.35
ELANE P08246 1/20 0.35
HSP90AB1 P08238 1/20 0.35
KCNH2 Q12809 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3991826 0.93 TLR8 (0.70) TLR8TLR7ADORA3ADORA2AADORA1
SCHEMBL3991913 0.90 TLR7 (0.51) TLR8TLR7ADORA3ADORA2AADORA1
SCHEMBL3992188 0.89 TLR8 (0.51) TLR8TLR7ADORA3ADORA2AADORA1
SCHEMBL3993609 0.86 TLR8 (0.57) TLR8TLR7ADORA3ADORA2AADORA1
SCHEMBL5507105 0.85 TLR8 (0.41) TLR8TLR7ADORA3ADORA2AADORA1
SCHEMBL5192462 0.85 TLR8 (0.41) TLR8TLR7ADORA3ADORA2AADORA1
SCHEMBL5571999 0.83 TLR8 (0.54) TLR8TLR7ADORA3ADORA2AADORA1
SCHEMBL3995270 0.83 TLR8 (0.60) TLR8TLR7
SCHEMBL3999203 0.82 ADORA3 (0.54) TLR8TLR7ADORA3ADORA2AADORA1
Hydrochloric Acid SCHEMBL3995835 0.82 TLR8 (0.53) TLR8TLR7ADORA3ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1863814-A1 1-SUBSTITUTED PYRAZOLO (3,4-C) RING COMPOUNDS AS MODULATORS OF CYTOKINE BIOSYNTHESIS FOR THE TREATMENT OF VIRAL INFECTIONS AND NEOPLASTIC DISEASES Coley Pharmaceutical Group, Inc. (US) 2007-12-12 EP disclosed
WO-2006107851-A1 1-SUBSTITUTED PYRAZOLO (3,4-C) RING COMPOUNDS AS MODULATORS OF CYTOKINE BIOSYNTHESIS FOR THE TREATMENT OF VIRAL INFECTIONS AND NEOPLASTIC DISEASES COLEY PHARMACEUTICAL GROUP, INC. (US) 2006-10-12 WO disclosed