Pyrrolidine

Pyrrolidine

SCHEMBL5194052

C1CCNC1.COc1ccc(-c2nnc(NC3CCN(Cc4ccc(C(=O)O)cc4)C(I)C3)c3cc(OC)ccc23)cc1

nearest known ligand 0.39

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 3/20 0.39
JAK1 P23458 3/20 0.39
TYK2 P29597 3/20 0.39
JAK3 P52333 3/20 0.39
LTA4H P09960 2/20 0.38
ALDH1A1 P00352 2/20 0.36
THRB P10828 1/20 0.36
HTT P42858 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
OPRM1 P35372 1/20 0.35
OPRK1 P41145 1/20 0.35
MMP13 P45452 2/20 0.35
HDAC3 O15379 4/20 0.35
HDAC4 P56524 4/20 0.35
HDAC1 Q13547 4/20 0.35
HDAC7 Q8WUI4 4/20 0.35
HDAC2 Q92769 4/20 0.35
HDAC10 Q969S8 4/20 0.35
HDAC11 Q96DB2 4/20 0.35
EHMT2 Q96KQ7 4/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pyrrolidine SCHEMBL4843645 0.88 ACHE (0.46) JAK2JAK1JAK3LTA4HHDAC3
SCHEMBL4839200 0.83 ACHE (0.51) LTA4HHDAC3HDAC4HDAC1HDAC7
SCHEMBL4843086 0.76 ACHE (0.51) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL4843614 0.76 ACHE (0.51) HDAC3HDAC4HDAC1HDAC7HDAC2
Hydrochloric Acid SCHEMBL4843163 0.76 ACHE (0.50) HDAC3HDAC4HDAC1HDAC7HDAC2
Hydrochloric Acid SCHEMBL4843091 0.75 ACHE (0.49) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL5196850 0.75 ACHE (0.58) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL4843635 0.74 ACHE (0.47) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL5195812 0.74 ALDH1A1 (0.54) ALDH1A1THRBHTTL3MBTL1HDAC3
SCHEMBL5193700 0.74 ACHE (0.56) HDAC3HDAC4HDAC1HDAC7HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1737840-B1 1-AMINO-PHTHALAZINE DERIVATIVES, THE PREPARATION AND THE THERAPEUTIC USE THEREOF SANOFI AVENTIS (FR) 2007-09-12 EP disclosed