SCHEMBL5195684

SCHEMBL5195684

CC(C)COC(=O)c1cccc(N)c1

nearest known ligand 0.67

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 9/20 0.67
ADRB1 P08588 9/20 0.67
ADRB3 P13945 9/20 0.67
ALDH1A1 P00352 3/20 0.53
TSHR P16473 1/20 0.53
CHRNB2 P17787 1/20 0.50
CHRNA4 P43681 1/20 0.50
JMJD6 Q6NYC1 1/20 0.48
PBRM1 Q86U86 1/20 0.46
PLA2G1B P04054 1/20 0.46
ATG4B Q9Y4P1 1/20 0.46
NPC1 O15118 1/20 0.44
MITF O75030 1/20 0.44
LMNA P02545 1/20 0.44
POLB P06746 1/20 0.44
KDM4E B2RXH2 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL109308 0.88 ALDH1A1 (0.61) ADRB2ADRB1ADRB3ALDH1A1TSHR
SCHEMBL9576615 0.85 ADRB2 (0.61) ADRB2ADRB1ADRB3ALDH1A1TSHR
SCHEMBL28280197 0.84 ADRB2 (0.56) ADRB2ADRB1ADRB3ALDH1A1TSHR
SCHEMBL3864388 0.83 ALDH1A1 (0.50) ADRB2ADRB1ADRB3ALDH1A1TSHR
SCHEMBL9576607 0.83 ADRB2 (0.58) ADRB2ADRB1ADRB3ALDH1A1TSHR
SCHEMBL6057072 0.82 ADRB2 (0.66) ADRB2ADRB1ADRB3ALDH1A1TSHR
SCHEMBL163932 0.82 ADRB2 (0.60) ADRB2ADRB1ADRB3ALDH1A1TSHR
SCHEMBL5164967 0.82 ALDH1A1 (0.54) ADRB2ADRB1ADRB3ALDH1A1TSHR
SCHEMBL163931 0.82 ALDH1A1 (0.54) ADRB2ADRB1ADRB3ALDH1A1TSHR
SCHEMBL10455395 0.82 ALDH1A1 (0.54) ADRB2ADRB1ADRB3ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170137407-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INFINITY PHARMACEUTICALS, INC. 2017-05-18 US disclosed
US-9546180-B2 Heterocyclic compounds and uses thereof INFINITY PHARMACEUTICALS, INC. (US) 2017-01-17 US disclosed
US-9115141-B2 Substituted isoquinolinones and methods of treatment thereof INFINITY PHARMACEUTICALS, INC. (US) 2015-08-25 US disclosed
US-20140288048-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INFINITY PHARMACEUTICALS, INC. 2014-09-25 US disclosed
US-8785470-B2 Heterocyclic compounds and uses thereof INFINITY PHARMACEUTICALS, INC. (US) 2014-07-22 US disclosed
EP-1812383-A1 GLYCOGEN PHOSPHORYLASE INHIBITOR COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF Smithkline Beecham Corporation (US) 2007-08-01 EP disclosed
WO-2006052722-A1 GLYCOGEN PHOSPHORYLASE INHIBITOR COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF SMITHKLINE BEECHAM CORPORATION (US) 2006-05-18 WO disclosed
US-4886813-A INHIBITORS OF ANGIOTENSIN CONVERTING ENZYME OTSUKA PHARMACEUTICAL FACTORY, INC. (JP) 1989-12-12 US disclosed
US-4379819-A OIL SOLUBLE MONOAZO DYE CIBA-GEIGY AG (CH) 1983-04-12 US disclosed
US-4080322-A WATER SOLUBLE DYES FOR LEATHER, PAPER, AND NON-WOVEN TEXTILES SANDOZ LTD. (CH) 1978-03-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140288048-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF AKT3, PIK3CA, AKT1 ADRB2 4048/4885ADRB1 3597/4885ADRB3 1196/4885
US-20170137407-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF AKT3, PIK3CA, AKT1 ADRB2 4048/4885ADRB1 3597/4885ADRB3 1196/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.