SCHEMBL5196325

SCHEMBL5196325

COc1ccc(CN2CCOC(C(N)=O)C2)cc1

nearest known ligand 0.64

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 8/20 0.64
SMN1; SMN2 Q16637 1/20 0.56
DRD2 P14416 1/20 0.56
DRD3 P35462 1/20 0.56
SIRT2 Q8IXJ6 1/20 0.53
SIRT1 Q96EB6 1/20 0.53
TSHR P16473 1/20 0.50
HIF1A Q16665 1/20 0.50
EPAS1 Q99814 1/20 0.50
GRIN2B Q13224 2/20 0.49
OPRM1 P35372 1/20 0.49
OPRK1 P41145 1/20 0.49
KDM4E B2RXH2 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5194021 0.88 SIGMAR1 (0.54) DRD4DRD2DRD3SIRT2SIRT1
SCHEMBL12696683 0.88 DRD4 (0.55) DRD4SMN1; SMN2GRIN2BKDM4E
SCHEMBL12696708 0.84 DRD4 (0.54) DRD4DRD2DRD3TSHRGRIN2B
SCHEMBL12696566 0.82 DRD4 (0.56) DRD4DRD2DRD3SIRT1GRIN2B
SCHEMBL2447401 0.82 DRD4 (0.56) DRD4DRD2DRD3SIRT1GRIN2B
SCHEMBL14357562 0.82 DRD4 (0.62) DRD4DRD2DRD3TSHRGRIN2B
SCHEMBL8329098 0.79 DRD4 (0.74) DRD4SMN1; SMN2DRD2DRD3
SCHEMBL20945053 0.79 DRD4 (0.74) DRD4SMN1; SMN2DRD2DRD3
SCHEMBL8327676 0.77 DRD4 (0.64) DRD4SMN1; SMN2DRD2DRD3TSHR
SCHEMBL14388375 0.77 DRD4 (0.62) DRD4DRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0968206-B8 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX INC (US) 2007-01-24 EP claimed
EP-0968206-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 2000-01-05 EP claimed
WO-1998037079-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 1998-08-27 WO claimed