SCHEMBL5196496

SCHEMBL5196496

CC(C)(C)[Si](C)(C)OCC#CCc1cc2ccccc2s1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AGXT P21549 1/20 0.46
CYP2A6 P11509 3/20 0.42
ADRB2 P07550 1/20 0.42
ASIC3 Q9UHC3 1/20 0.42
LOXL2 Q9Y4K0 1/20 0.42
ADRA1D P25100 2/20 0.36
CASR P41180 1/20 0.34
CA2 P00918 1/20 0.34
GLS O94925 2/20 0.33
IDH1 O75874 1/20 0.33
CHRNA7 P36544 1/20 0.33
MGLL Q99685 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4607947 0.70 BACE1 (0.32)
SCHEMBL8664580 0.70 HRH3 (0.35)
SCHEMBL662224 0.69 AGXT (0.43) AGXTCYP2A6ADRB2ASIC3LOXL2
SCHEMBL2168948 0.69
SCHEMBL1246811 0.68 PRKCI (0.33)
SCHEMBL660879 0.68 AGXT (0.42) AGXTCYP2A6ADRB2ASIC3LOXL2
SCHEMBL6844411 0.68 AGXT (0.42) AGXTCYP2A6ADRB2ASIC3LOXL2
SCHEMBL660878 0.68 AGXT (0.42) AGXTCYP2A6ADRB2ASIC3LOXL2
SCHEMBL274427 0.67 CYP2A6 (0.58) AGXTCYP2A6ADRB2ASIC3LOXL2
SCHEMBL347531 0.67 CYP2A6 (0.58) AGXTCYP2A6ADRB2ASIC3LOXL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1812387-A1 2,3,4-SUBSTITUTED CYCLOPENTANONES AS THERAPEUTIC AGENTS Allergan, Inc. (US) 2007-08-01 EP disclosed
WO-2006055481-A1 2,3,4-SUBSTITUTED CYCLOPENTANONES AS THERAPEUTIC AGENTS ALLERGAN , INC. (US) 2006-05-26 WO disclosed