SCHEMBL5196868

SCHEMBL5196868

CC(=CCC(C)N)c1cncc(OC2CCCCC2)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LNPEP Q9UIQ6 10/20 0.37
GRIN2D O15399 1/20 0.36
GRIN3B O60391 1/20 0.36
GRIN1 Q05586 1/20 0.36
GRIN2A Q12879 1/20 0.36
GRIN2B Q13224 1/20 0.36
GRIN2C Q14957 1/20 0.36
GRIN3A Q8TCU5 1/20 0.36
PDGFRB P09619 1/20 0.34
PDGFRA P16234 1/20 0.34
OPRK1 P41145 1/20 0.34
KCNH2 Q12809 1/20 0.34
PRMT5 O14744 1/20 0.34
CFTR P13569 1/20 0.34
CHRNB2 P17787 1/20 0.33
CHRNA4 P43681 1/20 0.33
MAP4K4 O95819 1/20 0.32
RIPK2 O43353 1/20 0.32
LOX P28300 1/20 0.32
LOXL2 Q9Y4K0 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL365734 0.80 MKNK2 (0.37) MAP4K4
SCHEMBL1691836 0.79 CHRNB2 (0.41) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL4242135 0.78 CHRNB2 (0.36) CHRNB2CHRNA4
SCHEMBL7529716 0.73 KDM4E (0.40)
SCHEMBL6453865 0.72 KDM4E (0.44)
SCHEMBL3931389 0.70 NPC1 (0.47) OPRK1KCNH2CHRNB2CHRNA4MAP4K4
SCHEMBL4422415 0.69 HCAR2 (0.32)
SCHEMBL7071083 0.68 MKNK2 (0.35) KCNH2MAP4K4
SCHEMBL5196864 0.67 CHRNB2 (0.41) LNPEPGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL5196862 0.67 CHRNB2 (0.41) LNPEPGRIN2DGRIN3BGRIN1GRIN2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1814852-A2 HYDROXYBENZOATE SALTS OF METANICOTINE COMPOUNDS Targacept, Inc. (US) 2007-08-08 EP disclosed
WO-2006053082-A2 HYDROXYBENZOATE SALTS OF METANICOTINE COMPOUNDS TARGACEPT, INC. (US) 2006-05-18 WO disclosed