SCHEMBL5196889

SCHEMBL5196889

Oc1cccc2c1Oc1cc(-c3cccnc3)ccc1N2C1CC2CCC(C1)N2CCc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 6/20 0.36
CYP11B2 P19099 6/20 0.36
HRH3 Q9Y5N1 1/20 0.35
GSK3B P49841 1/20 0.35
DRD2 P14416 2/20 0.35
DRD4 P21917 1/20 0.35
OPRM1 P35372 4/20 0.35
OPRD1 P41143 4/20 0.35
BRD4 O60885 1/20 0.34
CHRNA7 P36544 2/20 0.34
KCNH2 Q12809 2/20 0.34
HTR2A P28223 2/20 0.34
OPRK1 P41145 2/20 0.34
HTR2C P28335 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3167855 0.91 HRH3 (0.37) HRH3DRD2DRD4OPRM1OPRD1
SCHEMBL13395081 0.91 HRH3 (0.37) HRH3DRD2DRD4OPRM1OPRD1
SCHEMBL3177398 0.89 CYP11B1 (0.40) CYP11B1CYP11B2HRH3GSK3BDRD2
SCHEMBL13394862 0.89 CYP11B1 (0.40) CYP11B1CYP11B2HRH3GSK3BDRD2
SCHEMBL13394898 0.89 CYP11B1 (0.40) CYP11B1CYP11B2HRH3GSK3BDRD2
SCHEMBL5197806 0.88 HCRTR1 (0.39) CYP11B1CYP11B2HRH3DRD2DRD4
SCHEMBL13395065 0.85 OPRM1 (0.37) CYP11B1CYP11B2OPRM1BRD4KCNH2
SCHEMBL3173482 0.85 OPRM1 (0.37) CYP11B1CYP11B2OPRM1BRD4KCNH2
SCHEMBL4519661 0.82 HRH3 (0.35) CYP11B1CYP11B2HRH3GSK3BDRD2
SCHEMBL3188918 0.81 CYP11B2 (0.39) CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1833826-A2 TRICYCLIC DELTA-OPIOID MODULATORS JANSSEN PHARMACEUTICA N.V. (BE) 2007-09-19 EP disclosed
WO-2006069276-A2 TRICYCLIC ō-OPIOID MODULATORS JANSSEN PHARMACEUTICA N.V. (BE) 2006-06-29 WO disclosed